GRL 06579A (CID 9547976) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(5)
 
 
Top Targets:
HIV retropeps..(1)
 
 
BioAssay Types:
Literature(5)
 
 
BioActivity Types:
IC50(2)
 
 
Ki(1)
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103556843]
Ki 3.5e-06Inhibition of HIV1 protease dimerization in MT2 cells [AID328062, Type: Literature]
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2
[SID103556843]
IC50 0.0014Antiviral activity against HIV1 LAI in MT2 cells [AID328063, Type: Literature]
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3
[SID103556843]
IC50 0.0018Inhibition of HIV1 protease [AID311574, Type: Literature]
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4
[SID46394238]
 Experimentally measured binding affinity data derived from PDB [AID1811, Type: Literature]Chain A, Wild-Type Hiv-1 Protease In Complex With Potent Inhibitor Grl06579 [gi:114794303]
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5
[SID103556843]
 Inhibition of HIV1 protease dimerization in MT2 cells at 1 uM [AID328067, Type: Literature]
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