| 1 | [SID26747896] | Inactive | Potency | | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1: Spectroscopic Profiling in AFC Spectral Region [AID923, Type: confirmatory] | |  View X | Row No. | 1 | | Structure | 
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1: Spectroscopic Profiling in AFC Spectral Region | | AID | 923 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 2 | [SID26747896] | Inactive | Potency | | Counterscreen qHTS for Inhibitors of Tau Fibril Formation, Fluorescence Polarization [AID1463, Type: confirmatory] | | View X | Row No. | 2 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | Counterscreen qHTS for Inhibitors of Tau Fibril Formation, Fluorescence Polarization | | AID | 1463 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 3 | [SID26747896] | Inactive | Potency | | qHTS Assay for Compounds Blocking the Interaction Between CBF-beta and RUNX1 for the Treatment of Acute Myeloid Leukemia [AID1477, Type: confirmatory] | | View X | Row No. | 3 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Compounds Blocking the Interaction Between CBF-beta and RUNX1 for the Treatment of Acute Myeloid Leukemia | | AID | 1477 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 4 | [SID26747896] | Inactive | Potency | | qHTS Assay for Lipid Storage Modulators [AID1519, Type: confirmatory] | | View X | Row No. | 4 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Lipid Storage Modulators | | AID | 1519 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 5 | [SID26747896] | Inactive | Potency | | Quantitative High-Throughput Screen for Regulators of Epigenetic Control [AID1865, Type: confirmatory] | | View X | Row No. | 5 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | Quantitative High-Throughput Screen for Regulators of Epigenetic Control | | AID | 1865 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 6 | [SID26747896] | Inactive | Potency | | qHTS Assay for Compounds that Induce Erasure of Genomic Imprints [AID1948, Type: confirmatory] | | View X | Row No. | 6 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Compounds that Induce Erasure of Genomic Imprints | | AID | 1948 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 7 | [SID26747896] | Inactive | Potency | | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory] | | View X | Row No. | 7 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT | | AID | 686979 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 8 | [SID26747896] | Inactive | Potency | | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory] | | View X | Row No. | 8 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT | | AID | 686978 | | BioAssay type | confirmatory | | Target | | | PubMed | | | Data Table | |
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| 9 | [SID26747896] | Inactive | Potency | | Counterscreen for Luciferase (Kinase-Glo TM) Inhibition [AID1379, Type: confirmatory] | luciferase [Photuris pennsylvanica] [gi:1669525] | View X | Row No. | 9 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | Counterscreen for Luciferase (Kinase-Glo TM) Inhibition | | AID | 1379 | | BioAssay type | confirmatory | | Target | luciferase [Photuris pennsylvanica] [gi:1669525] | | PubMed | | | Data Table | |
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| 10 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1) [AID2517, Type: confirmatory] | Chain A, Human Ape1 Endonuclease With Bound Abasic Dna And Mn2+ Ion [gi:6980812] | View X | Row No. | 10 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of the Human Apurinic/apyrimidinic Endonuclease 1 (APE1) | | AID | 2517 | | BioAssay type | confirmatory | | Target | Chain A, Human Ape1 Endonuclease With Bound Abasic Dna And Mn2+ Ion [gi:6980812] | | PubMed | | | Data Table | |
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| 11 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase) [AID1490, Type: confirmatory] | phosphopantetheinyl transferase [Bacillus subtilis] [gi:10954339] | View X | Row No. | 11 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Bacillus subtilis Sfp phosphopantetheinyl transferase (PPTase) | | AID | 1490 | | BioAssay type | confirmatory | | Target | phosphopantetheinyl transferase [Bacillus subtilis] [gi:10954339] | | PubMed | | | Data Table | |
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| 12 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1) [AID485290, Type: confirmatory] | Chain A, Crystal Structure Of Human Tyrosyl-Dna Phosphodiesterase (Tdp1) [gi:20150581] | View X | Row No. | 12 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Tyrosyl-DNA Phosphodiesterase (TDP1) | | AID | 485290 | | BioAssay type | confirmatory | | Target | Chain A, Crystal Structure Of Human Tyrosyl-Dna Phosphodiesterase (Tdp1) [gi:20150581] | | PubMed | | | Data Table | |
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| 13 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia [AID2451, Type: confirmatory] | Chain A, Structure Of Giardia Fructose-1,6-Biphosphate Aldolase In Complex With Phosphoglycolohydrox [gi:122920737] | View X | Row No. | 13 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia | | AID | 2451 | | BioAssay type | confirmatory | | Target | Chain A, Structure Of Giardia Fructose-1,6-Biphosphate Aldolase In Complex With Phosphoglycolohydrox [gi:122920737] | | PubMed | | | Data Table | |
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| 14 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of HSD17B4, hydroxysteroid (17-beta) dehydrogenase 4 [AID893, Type: confirmatory] | Chain A, The Structure Of Wild-Type Human Hadh2 (17beta- Hydroxysteroid Dehydrogenase Type 10) Bound [gi:122921310] | View X | Row No. | 14 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of HSD17B4, hydroxysteroid (17-beta) dehydrogenase 4 | | AID | 893 | | BioAssay type | confirmatory | | Target | Chain A, The Structure Of Wild-Type Human Hadh2 (17beta- Hydroxysteroid Dehydrogenase Type 10) Bound [gi:122921310] | | PubMed | | | Data Table | |
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| 15 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of BRCT-Phosphoprotein Interaction (Red Fluorophore) [AID892, Type: confirmatory] | Chain A, Solution Structure Of The Brct-C Domain From Human Brca1 [gi:159162802] | View X | Row No. | 15 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of BRCT-Phosphoprotein Interaction (Red Fluorophore) | | AID | 892 | | BioAssay type | confirmatory | | Target | Chain A, Solution Structure Of The Brct-C Domain From Human Brca1 [gi:159162802] | | PubMed | | | Data Table | |
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| 16 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of BRCT-Phosphoprotein Interaction (Green Fluorophore) [AID875, Type: confirmatory] | Chain A, Solution Structure Of The Brct-C Domain From Human Brca1 [gi:159162802] | View X | Row No. | 16 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of BRCT-Phosphoprotein Interaction (Green Fluorophore) | | AID | 875 | | BioAssay type | confirmatory | | Target | Chain A, Solution Structure Of The Brct-C Domain From Human Brca1 [gi:159162802] | | PubMed | | | Data Table | |
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| 17 | [SID26747896] | Inactive | Potency | | qHTS for Inducers of the Endoplasmic Reticulum Stress Response (ERSR) in Human Glioma: qHTS [AID602332, Type: confirmatory] | heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) [Homo sapiens] [gi:168984549] | View X | Row No. | 17 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS for Inducers of the Endoplasmic Reticulum Stress Response (ERSR) in Human Glioma: qHTS | | AID | 602332 | | BioAssay type | confirmatory | | Target | heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) [Homo sapiens] [gi:168984549] | | PubMed | | | Data Table | |
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| 18 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory] | euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070] | View X | Row No. | 18 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a | | AID | 504332 | | BioAssay type | confirmatory | | Target | euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070] | | PubMed | | | Data Table | |
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| 19 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) [AID2147, Type: confirmatory] | Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486] | View X | Row No. | 19 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) | | AID | 2147 | | BioAssay type | confirmatory | | Target | Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486] | | PubMed | | | Data Table | |
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| 20 | [SID26747896] | Inactive | Potency | | qHTS Assay for Identification of Novel General Anesthetics [AID485281, Type: confirmatory] | Chain A, Horse Spleen Apoferritin [gi:254220970] | View X | Row No. | 20 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Identification of Novel General Anesthetics | | AID | 485281 | | BioAssay type | confirmatory | | Target | Chain A, Horse Spleen Apoferritin [gi:254220970] | | PubMed | | | Data Table | |
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| 21 | [SID26747896] | Inactive | Potency | | qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (without detergent) [AID1476, Type: confirmatory] | Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097] | View X | Row No. | 21 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (without detergent) | | AID | 1476 | | BioAssay type | confirmatory | | Target | Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097] | | PubMed | | | Data Table | |
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| 22 | [SID26747896] | Inactive | Potency | | qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (with detergent) [AID1478, Type: confirmatory] | Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097] | View X | Row No. | 22 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Promiscuous and Specific Inhibitors of Cruzain (with detergent) | | AID | 1478 | | BioAssay type | confirmatory | | Target | Chain A, Crystal Structure Of Cruzain Covalently Bound To A Purine Nitrile [gi:281307097] | | PubMed | | | Data Table | |
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| 23 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1) [AID2549, Type: confirmatory] | Chain A, Structure Of Human Recq-Like Helicase In Complex With A Dna Substrate [gi:282403581] | View X | Row No. | 23 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of RecQ-Like Dna Helicase 1 (RECQ1) | | AID | 2549 | | BioAssay type | confirmatory | | Target | Chain A, Structure Of Human Recq-Like Helicase In Complex With A Dna Substrate [gi:282403581] | | PubMed | | | Data Table | |
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| 24 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory] | aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681] | View X | Row No. | 24 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) | | AID | 1030 | | BioAssay type | confirmatory | | Target | aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681] | | PubMed | | | Data Table | |
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| 25 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) [AID1030, Type: confirmatory] | aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681] | View X | Row No. | 25 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Aldehyde Dehydrogenase 1 (ALDH1A1) | | AID | 1030 | | BioAssay type | confirmatory | | Target | aldehyde dehydrogenase 1 family, member A1 [Homo sapiens] [gi:30582681] | | PubMed | | | Data Table | |
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| 26 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of 12-hLO (12-human lipoxygenase) [AID1452, Type: confirmatory] | arachidonate 12-lipoxygenase, 12S-type [Homo sapiens] [gi:154426292] | View X | Row No. | 26 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of 12-hLO (12-human lipoxygenase) | | AID | 1452 | | BioAssay type | confirmatory | | Target | arachidonate 12-lipoxygenase, 12S-type [Homo sapiens] [gi:154426292] | | PubMed | | | Data Table | |
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| 27 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of 12-hLO (12-human lipoxygenase) [AID1452, Type: confirmatory] | arachidonate 12-lipoxygenase, 12S-type [Homo sapiens] [gi:154426292] | View X | Row No. | 27 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of 12-hLO (12-human lipoxygenase) | | AID | 1452 | | BioAssay type | confirmatory | | Target | arachidonate 12-lipoxygenase, 12S-type [Homo sapiens] [gi:154426292] | | PubMed | | | Data Table | |
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| 28 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of 15-hLO (15-human lipoxygenase) [AID887, Type: confirmatory] | 15-lipoxygenase [Homo sapiens] [gi:1832253] | View X | Row No. | 28 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of 15-hLO (15-human lipoxygenase) | | AID | 887 | | BioAssay type | confirmatory | | Target | 15-lipoxygenase [Homo sapiens] [gi:1832253] | | PubMed | | | Data Table | |
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| 29 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of 15-hLO (15-human lipoxygenase) [AID887, Type: confirmatory] | 15-lipoxygenase [Homo sapiens] [gi:1832253] | View X | Row No. | 29 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of 15-hLO (15-human lipoxygenase) | | AID | 887 | | BioAssay type | confirmatory | | Target | 15-lipoxygenase [Homo sapiens] [gi:1832253] | | PubMed | | | Data Table | |
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| 30 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of 15-hLO-2 (15-human lipoxygenase 2) [AID881, Type: confirmatory] | Arachidonate 15-lipoxygenase B [gi:317373425] | View X | Row No. | 30 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of 15-hLO-2 (15-human lipoxygenase 2) | | AID | 881 | | BioAssay type | confirmatory | | Target | Arachidonate 15-lipoxygenase B [gi:317373425] | | PubMed | | | Data Table | |
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| 31 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of Bloom's syndrome helicase (BLM) [AID2528, Type: confirmatory] | Bloom syndrome protein [Homo sapiens] [gi:4557365] | View X | Row No. | 31 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of Bloom's syndrome helicase (BLM) | | AID | 2528 | | BioAssay type | confirmatory | | Target | Bloom syndrome protein [Homo sapiens] [gi:4557365] | | PubMed | | | Data Table | |
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| 32 | [SID26747896] | Inactive | Potency | | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1 [AID900, Type: confirmatory] | caspase-1 isoform alpha precursor [Homo sapiens] [gi:15431328] | View X | Row No. | 32 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1 | | AID | 900 | | BioAssay type | confirmatory | | Target | caspase-1 isoform alpha precursor [Homo sapiens] [gi:15431328] | | PubMed | | | Data Table | |
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| 33 | [SID26747896] | Inactive | Potency | | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1 [AID900, Type: confirmatory] | caspase-1 isoform alpha precursor [Homo sapiens] [gi:15431328] | View X | Row No. | 33 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1 | | AID | 900 | | BioAssay type | confirmatory | | Target | caspase-1 isoform alpha precursor [Homo sapiens] [gi:15431328] | | PubMed | | | Data Table | |
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| 34 | [SID26747896] | Inactive | Potency | | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-7 [AID889, Type: confirmatory] | Caspase-7 [gi:1730092] | View X | Row No. | 34 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-7 | | AID | 889 | | BioAssay type | confirmatory | | Target | Caspase-7 [gi:1730092] | | PubMed | | | Data Table | |
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| 35 | [SID26747896] | Inactive | Potency | | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-7 [AID889, Type: confirmatory] | Caspase-7 [gi:1730092] | View X | Row No. | 35 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-7 | | AID | 889 | | BioAssay type | confirmatory | | Target | Caspase-7 [gi:1730092] | | PubMed | | | Data Table | |
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| 36 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory] | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | View X | Row No. | 36 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 | | AID | 884 | | BioAssay type | confirmatory | | Target | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | | PubMed | | | Data Table | |
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| 37 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory] | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | View X | Row No. | 37 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 | | AID | 884 | | BioAssay type | confirmatory | | Target | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | | PubMed | | | Data Table | |
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| 38 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory] | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | View X | Row No. | 38 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 | | AID | 884 | | BioAssay type | confirmatory | | Target | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | | PubMed | | | Data Table | |
|
| 39 | [SID26747896] | Inactive | Potency | | qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory] | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | View X | Row No. | 39 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Activators of Cytochrome P450 3A4 | | AID | 885 | | BioAssay type | confirmatory | | Target | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | | PubMed | | | Data Table | |
|
| 40 | [SID26747896] | Inactive | Potency | | qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory] | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | View X | Row No. | 40 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Activators of Cytochrome P450 3A4 | | AID | 885 | | BioAssay type | confirmatory | | Target | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | | PubMed | | | Data Table | |
|
| 41 | [SID26747896] | Inactive | Potency | | qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory] | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | View X | Row No. | 41 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Activators of Cytochrome P450 3A4 | | AID | 885 | | BioAssay type | confirmatory | | Target | cytochrome P450, family 3, subfamily A, polypeptide 4 [Homo sapiens] [gi:13435386] | | PubMed | | | Data Table | |
|
| 42 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate [AID2112, Type: confirmatory] | lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891] | View X | Row No. | 42 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate | | AID | 2112 | | BioAssay type | confirmatory | | Target | lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891] | | PubMed | | | Data Table | |
|
| 43 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate [AID2112, Type: confirmatory] | lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891] | View X | Row No. | 43 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate | | AID | 2112 | | BioAssay type | confirmatory | | Target | lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891] | | PubMed | | | Data Table | |
|
| 44 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate [AID2112, Type: confirmatory] | lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891] | View X | Row No. | 44 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Activators of Human alpha-Glucosidase From Spleen Homogenate | | AID | 2112 | | BioAssay type | confirmatory | | Target | lysosomal alpha-glucosidase preproprotein [Homo sapiens] [gi:119393891] | | PubMed | | | Data Table | |
|
| 45 | [SID26747896] | Inactive | | | qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen [AID2472, Type: screening] | glyceraldehyde-3-phosphate dehydrogenase [Homo sapiens] [gi:7669492] | View X | Row No. | 45 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | BioAssay | qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen | | AID | 2472 | | BioAssay type | screening | | Target | glyceraldehyde-3-phosphate dehydrogenase [Homo sapiens] [gi:7669492] | | PubMed | | | Data Table | |
|
| 46 | [SID26747896] | Inactive | | | qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen [AID2472, Type: screening] | glyceraldehyde-3-phosphate dehydrogenase [Homo sapiens] [gi:7669492] | View X | Row No. | 46 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | BioAssay | qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen | | AID | 2472 | | BioAssay type | screening | | Target | glyceraldehyde-3-phosphate dehydrogenase [Homo sapiens] [gi:7669492] | | PubMed | | | Data Table | |
|
| 47 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease [AID2101, Type: confirmatory] | glucocerebrosidase [Homo sapiens] [gi:496369] | View X | Row No. | 47 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease | | AID | 2101 | | BioAssay type | confirmatory | | Target | glucocerebrosidase [Homo sapiens] [gi:496369] | | PubMed | | | Data Table | |
|
| 48 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease [AID2101, Type: confirmatory] | glucocerebrosidase [Homo sapiens] [gi:496369] | View X | Row No. | 48 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors and Activators of N370S glucocerebrosidase as a Potential Chaperone Treatment of Gaucher Disease | | AID | 2101 | | BioAssay type | confirmatory | | Target | glucocerebrosidase [Homo sapiens] [gi:496369] | | PubMed | | | Data Table | |
|
| 49 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of GCN5L2 [AID504327, Type: confirmatory] | histone acetyltransferase KAT2A [Homo sapiens] [gi:153791535] | View X | Row No. | 49 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of GCN5L2 | | AID | 504327 | | BioAssay type | confirmatory | | Target | histone acetyltransferase KAT2A [Homo sapiens] [gi:153791535] | | PubMed | | | Data Table | |
|
| 50 | [SID26747896] | Inactive | Potency | | qHTS Assay for Inhibitors of GCN5L2 [AID504327, Type: confirmatory] | histone acetyltransferase KAT2A [Homo sapiens] [gi:153791535] | View X | Row No. | 50 | | Structure |
| | Substance | | | SID | 26747896 | | CID | 9543187 | | Outcome | Inactive | | Potency | [uM] | | BioAssay | qHTS Assay for Inhibitors of GCN5L2 | | AID | 504327 | | BioAssay type | confirmatory | | Target | histone acetyltransferase KAT2A [Homo sapiens] [gi:153791535] | | PubMed | | | Data Table | |
|
Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
