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imidacloprid (CID 86418) - Compound BioActivity Data
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BioActivity Outcomes:
Active(22)
 
 
Inactive(819)
 
 
Inconclusive(23)
 
 
Unspecified(26)
 
 
Top Targets:
NR LBD AR(23)
 
 
 
NR LBD ER(23)
 
 
NR LBD PPAR(23)
 
 
 
7TM GPCR Srx(21)
 
 
7TM GPCR Srsx(19)
 
 
BioAssay Types:
Confirmatory(391)
 
 
 
 
 
Screening(376)
 
 
 
 
Summary(63)
 
 
 
Literature(46)
 
 
 
 
BioActivity Types:
Potency(406)
 
 
 
 
 
IC50(31)
 
 
 
Ki(8)
 
 
EC50(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 648    Data Row: 890   Total Pages: 45   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103565844]
Ki 0.0019Binding affinity for nAChR with [3H]imidacloprid in Myzus persicae [AID147718, Type: Literature]
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2
[SID103565844]
Ki 0.0021Binding affinity for nAChR with [3H]imidacloprid in Drosophila [AID147717, Type: Literature]
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3
[SID103565844]
Ki 0.0022Potency to displace [3H]IMI binding to Nicotinic acetylcholine receptor from Drosophila head membranes [AID145345, Type: Literature]
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4
[SID103565844]
IC50 0.0036Displacement of [3H]IMI from peach-potato aphid alpha2/rat beta2 nAChR hybrid recombinant receptor [AID344086, Type: Literature]
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5
[SID103565844]
IC50 0.0043Displacement of [3H]IMI from nAChR in Drosophila brain [AID344082, Type: Literature]
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6
[SID103565844]
Ki 0.05Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranes [AID145520, Type: Literature]
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7
[SID103565844]
Ki 0.18Displacement of [3H]EPI from Aplysia AChBP expressed in HEK293S cells by scintillation proximity assay [AID318726, Type: Literature]
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8
[SID103565844]
Ki 0.267Displacement of [3H]ACE from Aplysia AChBP expressed in HEK293S cells by scintillation proximity assay [AID318725, Type: Literature]
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9
[SID103565844]
Ki 0.29Binding affinity for nAChR with [3H]nicotine in rat brain [AID145517, Type: Literature]
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10
[SID103565844]
Ki 0.72Potency to displace [3H]nicotine binding to Nicotinic acetylcholine receptor alpha4-beta2 immuno-isolated from M10 cells [AID146171, Type: Literature]
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11
[SID50086524]
Potency 1.122qHTS for Inhibitors of Cell Surface uPA Generation [AID540303, Type: confirmatory]urokinase-type plasminogen activator precursor [Mus musculus] [gi:6679377]
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12
[SID50086524]
Potency 1.122qHTS for Inhibitors of Cell Surface uPA Generation [AID540303, Type: confirmatory]urokinase plasminogen activator surface receptor precursor [Mus musculus] [gi:7242179]
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13
[SID50086524]
Potency 1.122qHTS for Inhibitors of Cell Surface uPA Generation [AID540303, Type: confirmatory]plasminogen precursor [Mus musculus] [gi:257471003]
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14
[SID50086524]
Potency 2.5929qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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15
[SID103565844]
IC50 2.6Displacement of [3H]nicotine from chick alpha4beta2 nAChR [AID344087, Type: Literature]Neuronal acetylcholine receptor subunit alpha-4 [gi:113062]
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16
[SID144206909]
Potency-Replicate_1 5.308qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line [AID743015, Type: confirmatory]
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17
[SID144206909]
Potency 6.6838qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in absence of CPT [AID686978, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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18
[SID144206909]
Potency-Replicate_1 8.4127qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line [AID743014, Type: confirmatory]
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19
[SID144206909]
Potency 8.4144qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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20
[SID50086524]
Potency 26.6795qHTS for Inhibitors of PLK1-PDB (polo-like kinase 1 - polo-box domain): Primary Screen [AID720504, Type: confirmatory]serine/threonine-protein kinase PLK1 [Homo sapiens] [gi:21359873]
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