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imidacloprid (CID 86418) - Compound BioActivity Data
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BioActivity Outcomes:
Active(121)
 
 
Inactive(609)
 
 
Inconclusive(15)
 
 
Unspecified(722)
 
 
Top Targets:
7tm 4(37)
 
 
Neur chan LBD(7)
 
 
 
NR LBD TR(6)
 
 
 
ANK(6)
 
 
 
Bromo ALL-1(5)
 
 
 
BioAssay Types:
Literature(760)
 
 
 
 
 
Screening(372)
 
 
 
 
Confirmatory(222)
 
 
 
 
 
BioActivity Types:
Potency(175)
 
 
 
 
 
IC50(52)
 
 
 
 
Ki(20)
 
 
 
EC50(7)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 1385    Data Row: 1467   Total Pages: 74   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103565844]
Ki 3.5e-05Displacement of [3H]-methyl-SFX from nAChR in Myzus persicae 4106A (green peach aphid) membrane after 70 min [AID1112903, Type: Literature]
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2
[SID103565844]
Ki 0.0019Binding affinity for nAChR with [3H]imidacloprid in Myzus persicae [AID147718, Type: Literature]
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3
[SID103565844]
Ki 0.0021Binding affinity for nAChR with [3H]imidacloprid in Drosophila [AID147717, Type: Literature]
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4
[SID103565844]
Ki 0.0022Potency to displace [3H]IMI binding to Nicotinic acetylcholine receptor from Drosophila head membranes [AID145345, Type: Literature]
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5
[SID103565844]
IC50 0.0023Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster head membrane after 90 min by filter binding assay [AID1101020, Type: Literature]Acetylcholine receptor subunit beta-like 2 [gi:14286096]
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6
[SID103565844]
IC50 0.0023Displacement of [3H]IMI from nicotinic acetylcholine receptor in Aphis craccivora (cowpea aphid) whole body membrane after 90 min by filter binding assay [AID1101022, Type: Literature]
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7
[SID103565844]
IC50 0.0026Displacement of [3H]IMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membrane after 90 min by filter binding assay [AID1101021, Type: Literature]
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8
[SID103565844]
Ki 0.003Displacement of [3H]IMI from nicotinic acetylcholine receptor in Drosophila melanogaster brain [AID1080614, Type: Literature]
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9
[SID103565844]
Ki 0.003Binding affinity to Drosophila brain nicotinic acetylcholine receptor assessed as [3H]IMI binding by radioligand binding assay [AID1092037, Type: Literature]
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10
[SID103565844]
IC50 0.0031Displacement of [3H]IMI from nicotinic acetylcholine receptor in Myzus persicae (green peach aphid) whole body membrane after 90 min by filter binding assay [AID1101023, Type: Literature]
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11
[SID103565844]
IC50 0.0036Displacement of [3H]IMI from peach-potato aphid alpha2/rat beta2 nAChR hybrid recombinant receptor [AID344086, Type: Literature]
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12
[SID103565844]
IC50 0.0043Displacement of [3H]IMI from nAChR in Drosophila brain [AID344082, Type: Literature]
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13
[SID103565844]
IC50 0.0046Inhibition of [3H]IMI binding to Drosophila melanogaster neuronal acetylcholine receptor [AID1101298, Type: Literature]Acetylcholine receptor subunit beta-like 2 [gi:14286096]
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14
[SID103565844]
Ki 0.0046Displacement of [3H]IMI from Musca domestica (house fly) brain nicotinic acetylcholine receptor [AID1091970, Type: Literature]
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15
[SID103565844]
Ki 0.019Binding affinity to salt water mollusc Aplysia californica AChBP Y55W mutant assessed as [3H]acetamiprid binding by radioligand binding assay [AID1092035, Type: Literature]Soluble acetylcholine receptor [gi:74820297]
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16
[SID103565844]
IC50 0.01995Displacement of [3H]imidacloprid from Musca domestica (house fly)-head membrane nAChR [AID1110486, Type: confirmatory]
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17
[SID103565844]
IC50 0.02Displacement of [3H]imidacloprid from Musca domestica (house fly)-head membrane nAChR [AID1110017, Type: confirmatory]
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18
[SID103565844]
IC50 0.02Displacement of [3HIMI from nicotinic acetylcholine receptor in Musca domestica (house fly) head membranes incubated for 60 min by liquid scintillation counting method [AID1102410, Type: Literature]
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19
[SID103565844]
Ki 0.032Displacement of [3H]IMD from nAChR in Myzus persicae 4106A (green peach aphid) membrane after 70 min [AID1112902, Type: Literature]
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20
[SID103565844]
Ki 0.05Binding affinity for nAChR with [3H]-nicotine in rat alpha4 beta2 membranes [AID145520, Type: Literature]
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