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Dimethoxyphenylethylamine (CID 8421) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Inactive(592)
 
 
Inconclusive(10)
 
 
Unspecified(9)
 
 
Top Targets:
7tm 4(37)
 
 
G-alpha(8)
 
 
 
Tryp SPc(7)
 
 
CAP ED(5)
 
 
TRP 2(5)
 
 
BioAssay Types:
Screening(391)
 
 
 
Confirmatory(180)
 
 
 
 
Literature(22)
 
 
 
 
 
BioActivity Types:
Potency(133)
 
 
 
 
IC50(35)
 
 
EC50(6)
 
 
Kd(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 555    Data Row: 613   Total Pages: 31   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103197783]
Kd 4.36516Affinity against 5-hydroxytryptamine receptors in rat fundus model [AID6406, Type: Literature]
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2
[SID14719304]
Aqueous Solubility from MLSMR Stock Solutions [AID1996, Type: other]
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3
[SID14719304]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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4
[SID103197783]
Log value of hallucinogenic activity was determined [AID19263, Type: Literature]
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5
[SID103197783]
Hallucinogenic activity i.e; ratio of effective dose of mescaline to the effective dose in human [AID88883, Type: Literature]
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6
[SID103197783]
Compound was tested for the psychotropic effect in human (activity is expressed in mescaline unit) [AID89086, Type: Literature]
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7
[SID103197783]
In vitro bovine plasma monoamine oxidase deamination with semicarbazide [AID125220, Type: Literature]
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8
[SID103197783]
In vitro bovine plasma monoamine oxidase deamination without semicarbazide [AID125221, Type: Literature]
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9
[SID103197783]
Antibacterial activity against Escherichia coli MG1655 overexpressing lolA assessed as growth inhibition after 16 hrs [AID743654, Type: Literature]
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10
[SID103197783]
Activity of human SSAO measured as hydrogen peroxide production at 1 mM relative to benzylamine oxidation [AID273097, Type: Literature]Membrane primary amine oxidase [gi:2501336]
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11
[SID103197783]
Activity of mouse SSAO measured as hydrogen peroxide production at 100 uM relative to benzylamine oxidation [AID273098, Type: Literature]Membrane primary amine oxidase [gi:5902787]
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12
[SID14719304]
Potency 11.2202qHTS Assay for Identification of Novel General Anesthetics [AID485281, Type: confirmatory]Chain A, Horse Spleen Apoferritin [gi:254220970]
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13
[SID14719304]
Potency 12.5893qHTS Assay for Identifying a Potential Treatment of Ataxia-Telangiectasia [AID485349, Type: confirmatory]serine-protein kinase ATM [Homo sapiens] [gi:71902540]
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14
[SID14719304]
Potency 39.8107qHTS Assay for Inhibitors of Human Jumonji Domain Containing 2E (JMJD2E) [AID2147, Type: confirmatory]Chain A, Crystal Structure Of The Human 2-Oxoglutarate Oxygenase Loc390245 [gi:221046486]
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15
[SID14719304]
Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the orexin 1 receptor (OX1R; HCRTR1) [AID434989, Type: screening]orexin receptor type 1 [Homo sapiens] [gi:222080095]
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16
[SID14719304]
FRET-based cell-based primary high throughput screening assay to identify antagonists of the orexin 1 receptor (OX1R; HCRTR1) [AID485270, Type: screening]orexin receptor type 1 [Homo sapiens] [gi:222080095]
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17
[SID14719304]
Fluorescence-based biochemical high throughput primary assay to identify inhibitors of phospholipase C isozymes (PLC-gamma1). [AID720700, Type: screening]Phospholipase C, gamma 1 [Homo sapiens] [gi:223459640]
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18
[SID14719304]
Potency Nrf2 qHTS screen for inhibitors [AID504444, Type: confirmatory]nuclear factor erythroid 2-related factor 2 isoform 2 [Homo sapiens] [gi:224028257]
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19
[SID14719304]
Fluorescence polarization to screen for inhibitors that disrupt the protein-protein interaction between Keap1 and Nrf2 Measured in Biochemical System Using Plate Reader - 2119-01_Inhibitor_SinglePoint_HTS_Activity [AID504523, Type: screening]nuclear factor erythroid 2-related factor 2 isoform 2 [Homo sapiens] [gi:224028257]
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20
[SID14719304]
uHTS identification of Caspase-8 TRAIL sensitizers in a luminesence assay [AID624354, Type: screening]tumor necrosis factor receptor superfamily member 10B isoform 1 precursor [Homo sapiens] [gi:224494019]
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