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lomatin (CID 759302) - Compound BioActivity Data
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BioActivity Outcomes:
Active(7)
 
 
Inactive(590)
 
 
Inconclusive(8)
 
 
Unspecified(5)
 
 
Top Targets:
7TM GPCR Srx(21)
 
 
7TM GPCR Srsx(15)
 
 
G-alpha(8)
 
 
 
Tryp SPc(7)
 
 
Bcl-2 like(6)
 
 
 
BioAssay Types:
Screening(405)
 
 
 
 
Confirmatory(182)
 
 
 
 
Literature(17)
 
 
 
 
BioActivity Types:
Potency(134)
 
 
 
 
IC50(40)
 
 
 
EC50(5)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 550    Data Row: 610   Total Pages: 31   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID49646623]
Counterscreen for inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis: Fluroescence-based biochemical high throughput Glycerophosphate Dehydrogenase-Triosephosphate Isomerase (GDH-TPI) assay to identify assay artifacts [AID652141, Type: screening]
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2
[SID26725216]
uHTS of Mcl-1/Bid interaction inhibitors [AID1021, Type: screening]Mcl-1 [Homo sapiens] [gi:7582271]
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3
[SID49646623]
Fluorescence-based biochemical primary high throughput screening assay to identify inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis [AID588726, Type: screening]fructose-bisphosphate aldolase [Mycobacterium tuberculosis H37Rv] [gi:15607504]
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4
[SID49646623]
Fluorescence-based biochemical high throughput confirmation assay for inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis [AID651616, Type: screening]fructose-bisphosphate aldolase [Mycobacterium tuberculosis H37Rv] [gi:15607504]
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5
[SID103600440]
Binding affinity to spinach calmodulin assessed as modification of electrophoretic mobility at 0.033 ug/mL after 1.5 hrs by SDS-PAGE in presence of calcium chloride [AID334851, Type: Literature]Calmodulin [gi:122063217]
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6
[SID49646623]
Flow Cytometric HTS Screen for inhibitors of the ABC transporter ABCB6 for MLPCN Compound Set [AID602162, Type: screening]ATP-binding cassette sub-family B member 6, mitochondrial [Homo sapiens] [gi:9955963]
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7
[SID103600440]
Binding affinity to bovine brain calmodulin assessed as modification of electrophoretic mobility at 0.033 ug/mL after 1.5 hrs by SDS-PAGE in presence of calcium chloride [AID334850, Type: Literature]Calmodulin [gi:49037473]
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8
[SID103600440]
IC50 296Phytotoxicity against Echinochloa crus-galli assessed as inhibition of radicle elongation by petri dish bioassay [AID334617, Type: Literature]
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9
[SID103600440]
IC50 344Phytotoxicity against Amaranthus hypochondriacus assessed as inhibition of radicle elongation by petri dish bioassay [AID334616, Type: Literature]
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10
[SID103600440]
IC50 500Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate after 60 mins by fluorescence quenching assay [AID637774, Type: Literature]Beta-secretase 1 [gi:296434407]
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11
[SID103600440]
Inhibition of recombinant human BACE1 using Rh-EVNLDAEFK as substrate at 500 uM after 60 mins by fluorescence quenching assay [AID637775, Type: Literature]Beta-secretase 1 [gi:296434407]
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12
[SID49646623]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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13
[SID26725216]
Potency 4.4668qHTS Assay for Inhibitors of Influenza NS1 Protein Function [AID2326, Type: confirmatory]nonstructural protein 1 [Influenza A virus (A/WSN/1933(H1N1))] [gi:194352380]
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14
[SID26725216]
Potency 10.4179Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 96 hour incubation [AID504834, Type: confirmatory]
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15
[SID49646623]
Potency 11.2202qHTS for Agonist of gsp, the Etiologic Mutation Responsible for Fibrous Dysplasia/McCune-Albright Syndrome: qHTS [AID624287, Type: confirmatory]Guanine nucleotide-binding protein G(s) subunit alpha isoforms short [gi:52000961]
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16
[SID26725216]
Potency 11.6891Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation [AID504832, Type: confirmatory]
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17
[SID49646623]
Potency 22.3872qHTS Assay for Substrates of Mammalian Selenoprotein Thioredoxin Reductase 1 (TrxR1): qHTS [AID588456, Type: confirmatory]thioredoxin reductase [Rattus norvegicus] [gi:8659577]
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18
[SID26725216]
Absolute IC50 54Dose Response Confirmation for Mcl-1/Bid Interaction Inhibitors [AID1418, Type: confirmatory]Mcl-1 [Homo sapiens] [gi:7582271]
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19
[SID49646623]
uHTS identification of small molecule inhibitors of the catalytic domain of the SUMO protease, SENP1 in a FRET assay [AID624204, Type: screening]sentrin-specific protease 1 [Homo sapiens] [gi:7657550]
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20
[SID26725216]
qHTS Assay for Inhibitors of Fructose-1,6-bisphosphate Aldolase from Giardia Lamblia: Coupling assay counterscreen [AID2472, Type: screening]glyceraldehyde-3-phosphate dehydrogenase isoform 1 [Homo sapiens] [gi:7669492]
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