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benzylamine (CID 7504) - Compound BioActivity Data
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BioActivity Outcomes:
Active(16)
 
 
Inactive(135)
 
 
Inconclusive(2)
 
 
Unspecified(53)
 
 
Top Targets:
NR LBD PPAR(8)
 
 
Tryp SPc(7)
 
 
NR LBD ER(7)
 
 
NAD binding 8(7)
 
 
NR LBD AR(7)
 
 
 
BioAssay Types:
Confirmatory(87)
 
 
 
Literature(68)
 
 
 
 
Summary(24)
 
 
Screening(17)
 
 
BioActivity Types:
Potency(105)
 
 
 
Ki(10)
 
 
 
Kd(2)
 
 
IC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 196    Data Row: 206   Total Pages: 11   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103174520]
Km 6.7Michaelis-Menten constant for semicarbazide-sensitive amine oxidase (SSAO) from human, rat or mouse crude membranes [AID239765, Type: Literature]
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2
[SID103174520]
Km 15.4Binding affinity to mouse SSAO [AID273100, Type: Literature]Membrane primary amine oxidase [gi:5902787]
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3
[SID103174520]
Ki 20Displacement of [3H]clonidine from adrenergic alpha-1 receptor in Sprague-Dawley rat cortex [AID313559, Type: Literature]
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4
[SID103174520]
Ki 20In vitro for binding affinity against Alpha-2 adrenergic receptor by radioligand [3H]clonidine in rat [AID37364, Type: Literature]Alpha-2A adrenergic receptor [gi:231461]
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5
[SID103174520]
Ki 20In vitro for binding affinity against Alpha-2 adrenergic receptor by radioligand [3H]clonidine in rat [AID37364, Type: Literature]Alpha-2C adrenergic receptor [gi:231464]
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6
[SID103174520]
Ki 20In vitro for binding affinity against Alpha-2 adrenergic receptor by radioligand [3H]clonidine in rat [AID37364, Type: Literature]Alpha-2B adrenergic receptor [gi:47117345]
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7
[SID46393333]
Kd 144Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Trypsin Specificity As Elucidated By Lie Calculations, X-Ray Structures And Association Constant Measurements [gi:42543832]
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8
[SID46393336]
Kd 321Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Trypsin Specificity As Elucidated By Lie Calculations, X-Ray Structures And Association Constant Measurements [gi:42543836]
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9
[SID46393946]
Ki 1580Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB [AID977610, Type: Literature]Chain A, Bovine Pancreas Beta-Trypsin In Complex With Benzylamine [gi:4699788]
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10
[SID46393946]
Ki 1580Experimentally measured binding affinity data (Ki) for protein-ligand complexes derived from PDB [AID977610, Type: Literature]Chain A, Bovine Pancreas Beta-Trypsin In Complex With Benzylamine [gi:4699788]
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11
[SID46393333]
Experimentally measured binding affinity data derived from PDB [AID1811, Type: other]Chain A, Trypsin Specificity As Elucidated By Lie Calculations, X-Ray Structures And Association Constant Measurements [gi:42543832]
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12
[SID46393336]
Experimentally measured binding affinity data derived from PDB [AID1811, Type: other]Chain A, Trypsin Specificity As Elucidated By Lie Calculations, X-Ray Structures And Association Constant Measurements [gi:42543836]
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13
[SID46393946]
Experimentally measured binding affinity data derived from PDB [AID1811, Type: Literature]Chain A, Bovine Pancreas Beta-Trypsin In Complex With Benzylamine [gi:4699788]
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14
[SID103174520]
Stimulation of glucose transport in mouse adipocytes at 0.1 mM in presence of sodium orthovanadate [AID273101, Type: Literature]
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15
[SID103174520]
Stimulation of glucose transport in mouse adipocytes at 1 mM in presence of sodium orthovanadate [AID273102, Type: Literature]
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16
[SID48415031]
DSSTox (EPAFHM) EPA Fathead Minnow Acute Toxicity [AID1188, Type: other]
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17
[SID103174520]
IC50 40Antiproliferative activity against human SKBR3 cells after 72 hrs [AID304707, Type: Literature]
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18
[SID103174520]
Km 124Km for Benzylamine oxidase of porcine serum [AID239730, Type: Literature]
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19
[SID103174520]
Km 168.83Kinetic constant (Km) determined in rat brain mitochondria [AID125407, Type: Literature]
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20
[SID103174520]
Ki 170Inhibition of bovine PNMT by radiochemical assay [AID313558, Type: Literature]Phenylethanolamine N-methyltransferase [gi:130374]
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