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dipivefrin (CID 71486) - Compound BioActivity Data
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BioActivity Outcomes:
Active(21)
 
 
Inactive(487)
 
 
Inconclusive(21)
 
 
Unspecified(1)
 
 
Top Targets:
7tm 4(49)
 
 
 
 
NR LBD AR(7)
 
 
NR LBD ER(7)
 
 
Esterase lipa..(5)
 
 
PLDc mTdp1 2(4)
 
 
 
 
BioAssay Types:
Screening(319)
 
 
 
 
Confirmatory(164)
 
 
 
 
 
Summary(15)
 
 
 
Literature(13)
 
 
BioActivity Types:
Potency(164)
 
 
 
 
 
IC50(11)
 
 
EC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 476    Data Row: 530   Total Pages: 27   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID56463529]
Potency 0.2593qHTS assay of beta-arrestin-biased ligands of beta2-adrenergic receptor: Hit Validation with GloSensor [AID588790, Type: confirmatory]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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2
[SID56463529]
EC50_MICROM 7.13Dose response for HTS for Beta-2AR agonists via FAP method from CP1 [AID588763, Type: confirmatory]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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3
[SID144204226]
Potency 9.0349qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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4
[SID144204226]
Potency-Replicate_1 12.7448qHTS assay to identify small molecule antagonists of the thyroid receptor (TR) signaling pathway - cell viability counter screen [AID743064, Type: confirmatory]
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5
[SID144204226]
Potency-Replicate_1 12.7448qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - wild type cell line [AID743012, Type: confirmatory]
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6
[SID56463529]
Counterscreen for antagonists of the galanin Receptor 3 (GalR3): Fluorescence-based cell-based high throughput screening assay to identify non specific agonists of the parental HEK-CNG cells [AID652268, Type: screening]
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7
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Beta-3 adrenergic receptor [gi:461604]
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8
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Alpha-1D adrenergic receptor [gi:1168243]
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9
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Alpha-1A adrenergic receptor [gi:1168246]
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10
[SID56463529]
Fluorescence-based cell-based primary high throughput screening assay to identify antagonists of the Galanin Receptor 3 (GalR3) [AID651719, Type: screening]galanin receptor type 3 [Homo sapiens] [gi:4503907]
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11
[SID56463529]
Fluorescence-based cell-based primary high throughput confirmation assay to identify antagonists of the Galanin Receptor 3 (GalR3) [AID652245, Type: screening]galanin receptor type 3 [Homo sapiens] [gi:4503907]
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12
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Alpha-2A adrenergic receptor [gi:1351829]
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13
[SID56463529]
HTS for Beta-2AR agonists via FAP method, Single Point, Cherry Pick 1 [AID540358, Type: other]beta-2 adrenergic receptor [Homo sapiens] [gi:4501969]
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14
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Beta-1 adrenergic receptor [gi:48429211]
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15
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Alpha-2C adrenergic receptor [gi:20141211]
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16
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Alpha-1B adrenergic receptor [gi:116241241]
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17
[SID56463529]
qHTS of D3 Dopamine Receptor Potentiators: qHTS [AID652051, Type: screening]D(3) dopamine receptor isoform e [Homo sapiens] [gi:89191863]
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18
[SID56463529]
qHTS of D3 Dopamine Receptor Agonist: qHTS [AID652048, Type: screening]D(3) dopamine receptor isoform e [Homo sapiens] [gi:89191863]
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19
[SID103770816]
Adrenergic receptor agonist [AID742741, Type: other]Alpha-2B adrenergic receptor [gi:613504690]
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20
[SID56463529]
Fluorescence polarization-based primary biochemical high throughput screening assay to identify inhibitors of human platelet-activating factor acetylhydrolase 1b, catalytic subunit 2 (PAFAH1B2) [AID492953, Type: screening]platelet-activating factor acetylhydrolase IB subunit beta isoform b [Homo sapiens] [gi:296080766]
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