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CHEMBL2172448 (CID 71453585) - Compound BioActivity Data
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BioActivity Outcomes:
Unspecified(11)
 
 
Top Targets:
Lipase 3(7)
 
 
Amidase(1)
 
 
Hydrolase 4(1)
 
 
BioAssay Types:
Literature(11)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 11    Data Row: 11   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID163321230]
Inhibition of porcine pancreatic lipase type 2 at 10 uM by FRET assay [AID703150, Type: Literature]
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2
[SID163321230]
Inhibition of bacterial lipoprotein lipase at 10 uM by FRET assay [AID703152, Type: Literature]
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3
[SID163321230]
Inhibition of human DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 10 uM in detergent free solution by FRET assay [AID703154, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:114149271]
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4
[SID163321230]
Inhibition of mouse DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 10000 nM by scintillation counting based radio-TLC assay [AID703155, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:341940439]
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5
[SID163321230]
Inhibition of mouse DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 1000 nM by scintillation counting based radio-TLC assay [AID703156, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:341940439]
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6
[SID163321230]
Inhibition of mouse DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 100 nM by scintillation counting based radio-TLC assay [AID703157, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:341940439]
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7
[SID163321230]
Inhibition of mouse DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 10 nM by scintillation counting based radio-TLC assay [AID703158, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:341940439]
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8
[SID163321230]
Inhibition of human N-terminal histidine tagged full length MAGL expressed in Escherichia coli at 10 uM by by coumarin ester substrate fluorescence assay [AID703162, Type: Literature]Monoglyceride lipase [gi:47117287]
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9
[SID163321230]
Inhibition of rat histidine tagged FAAH expressed in Escherichia coli at 10 uM by coumarin ester substrate fluorescence assay [AID703165, Type: Literature]Fatty-acid amide hydrolase 1 [gi:6225312]
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10
[SID163321230]
Inhibition of human DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 10 uM in presence of 0.05% Triton X-100 by scintillation counting based radio-TLC assay [AID703168, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:114149271]
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11
[SID163321230]
Inhibition of human DAGLalpha expressed in HEK293T cell membrane using [14C]SAG substrate at 10 uM in presence of 0.05% Triton X-100 by FRET assay [AID703172, Type: Literature]Sn1-specific diacylglycerol lipase alpha [gi:114149271]
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