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CHEMBL2113575 (CID 71450937) - Compound BioActivity Data
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BioActivity Outcomes:
Active(1)
 
 
Unspecified(8)
 
 
Top Targets:
7tm 4(6)
 
 
 
BioAssay Types:
Literature(9)
 
 
 
BioActivity Types:
Ki(3)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 9   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID163316064]
Ki 0.021Affinity for adenosine A1 receptor of calf brain using 1 nM [3H]PIA [AID31978, Type: Literature]Adenosine receptor A1 [gi:160332359]
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2
[SID163316064]
Ki 60Affinity for adenosine A2 receptor at rat striatal membrane using 5 nM [3H]CGS-21680 [AID33430, Type: Literature]Adenosine receptor A2a [gi:8928539]
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3
[SID163316064]
Ki 60Affinity for adenosine A2 receptor at rat striatal membrane using 5 nM [3H]CGS-21680 [AID33430, Type: Literature]Adenosine receptor A2b [gi:112939]
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4
[SID163316064]
Selectivity ratio of compounds 9a and 9b against A2 receptor [AID232734, Type: Literature]Adenosine receptor A2b [gi:112939]
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5
[SID163316064]
Selectivity ratio of compounds 9a and 9b against A1 receptor [AID232733, Type: Literature]Adenosine receptor A1 [gi:2827766]
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6
[SID163316064]
Selectivity as ratio of Ki for binding to adenosine A1 and A2 receptors [AID32641, Type: Literature]Adenosine receptor A1 [gi:2827766]
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7
[SID163316064]
Selectivity as ratio of Ki for binding to adenosine A1 and A2 receptors [AID32641, Type: Literature]Adenosine receptor A2a [gi:8928539]
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8
[SID163316064]
Selectivity ratio of compounds 9a and 9b against A2 receptor [AID232734, Type: Literature]Adenosine receptor A2a [gi:8928539]
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9
[SID163316064]
Selectivity as ratio of Ki for binding to adenosine A1 and A2 receptors [AID32641, Type: Literature]Adenosine receptor A2b [gi:112939]
View