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CHEMBL2387140 (CID 71305062) - Compound BioActivity Data
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BioActivity Outcomes:
Active(4)
 
 
Unspecified(5)
 
 
Top Targets:
HDc(2)
 
 
BioAssay Types:
Literature(9)
 
 
 
BioActivity Types:
IC50(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 9    Data Row: 9   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID174486234]
IC50 0.045Inhibition of PDE2 (unknown origin) [AID748841, Type: Literature]
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2
[SID174486234]
IC50 0.045Inhibition of PDE2 catalytic domain (unknown origin) [AID749038, Type: Literature]
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3
[SID174486234]
IC50 0.378Inhibition of PDE4B (unknown origin) [AID748847, Type: Literature]cAMP-specific 3',5'-cyclic phosphodiesterase 4B [gi:729163]
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4
[SID174486234]
IC50 0.378Inhibition of PDE4B catalytic domain (unknown origin) [AID749039, Type: Literature]cAMP-specific 3',5'-cyclic phosphodiesterase 4B [gi:729163]
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5
[SID174486234]
Metabolic stability in human liver microsome assessed as half life [AID748839, Type: Literature]
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6
[SID174486234]
Selectivity ratio of IC50 for PDE4B (unknown origin) to IC50 for PDE2 (unknown origin) [AID748840, Type: Literature]
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7
[SID174486234]
Selectivity ratio of IC50 for PDE (unknown origin) to IC50 for PDE2 catalytic domain (unknown origin) [AID749016, Type: Literature]
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8
[SID174486234]
Half life in human liver microsomes [AID749035, Type: Literature]
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9
[SID174486234]
Selectivity ratio of IC50 for PDE4 (unknown origin) to IC50 for PDE2 catalytic domain (unknown origin) [AID749037, Type: Literature]
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