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CHEMBL2089186 (CID 70691263) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Top Targets:
PBP1 mGluR gr..(2)
 
 
BioAssay Types:
Literature(2)
 
 
BioActivity Types:
IC50(1)
 
 
Ki(1)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 2    Data Row: 2   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID160692035]
Ki 0.041Displacement of [3H]MPEP from mGluR5 in Sprague-Dawley rat brain membrane after 60 mins by liquid scintillation counting [AID683163, Type: Literature]Metabotropic glutamate receptor 5 [gi:1170947]
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2
[SID160692035]
IC50 0.08Inverse agonist activity at rat mGluR5 expressed in HEK293A cells coexpressing Gqalpha assessed as inhibition of quisqualic-induced D-myo-inositol 1 production by ELISA [AID683165, Type: Literature]Metabotropic glutamate receptor 5 [gi:1170947]
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