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[3H]-MLA (CID 70684997) - Compound BioActivity Data
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BioActivity Outcomes:
Active(4)
 
 
Unspecified(7)
 
 
Top Targets:
Neur chan LBD(3)
 
 
BioAssay Types:
Literature(8)
 
 
 
BioActivity Types:
Kd(4)
 
 
 
Ki(4)
 
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 10    Data Row: 11   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID160676124]
Ki 0.00098Inhibition of [3H]MLA binding in presence of methylcaconitine. [AID146953, Type: Literature]
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2
[SID160676124]
Ki 0.00178Inhibition of [3H]MLA binding in presence of alpha-bungarotoxin [AID146951, Type: Literature]
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3
[SID160676124]
Kd 0.0019Affinity constant Kd(nM) in rat brain cerebral cortex homogenates. [AID227640, Type: Literature]
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4
[SID160676124]
Ki 6.07Inhibition of [3H]MLA binding in presence of (-)-nicotine [AID146950, Type: Literature]
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5
[SID160676124]
Kd 0.0019GRAC: rat AChR-alpha7 radioligand [AID540485, Type: other]Neuronal acetylcholine receptor subunit alpha-7 [gi:146345356]
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6
[SID160676124]
Kd 0.0075GRAC: human AChR-alpha9-alpha10 radioligand [AID540743, Type: other]Neuronal acetylcholine receptor subunit alpha-9 [gi:308153406]
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7
[SID160676124]
Kd 0.0075GRAC: human AChR-alpha9-alpha10 radioligand [AID540743, Type: other]Neuronal acetylcholine receptor subunit alpha-10 [gi:14916526]
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8
[SID160676124]
Ki 20Inhibition of [3H]MLA binding in presence of mecamylamine [AID146952, Type: Literature]
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9
[SID160676124]
Inhibition of [125I]iodo-MLA binding in presence of 3-cinnamylidene-anabasine; ND means no data [AID146958, Type: Literature]
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10
[SID160676124]
Inhibition of [125I]iodo-MLA binding in presence of dihydro-beta-erythroidine; ND means no data [AID146959, Type: Literature]
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11
[SID160676124]
Bmax value(fmol/mg protein) was evaluated in rat brain using [125I]- alpha-BGT [AID227635, Type: Literature]
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