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CHEMBL2029000 (CID 70683606) - Compound BioActivity Data
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BioActivity Outcomes:
Active(4)
 
 
Inactive(4)
 
 
BioAssay Types:
Literature(8)
 
 
 
BioActivity Types:
EC50(5)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID160673019]
EC50 0.8Activity against human P2Y1-GFP expressed in 1321N1 cells by intracellular calcium increase [AID261698, Type: Literature]P2Y purinoceptor 1 [gi:1352692]
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2
[SID160673019]
Stability of the compound assessed as human e-NPP1-mediated hydrolysis at pH 8.5 after 20 mins by HPLC analysis [AID644880, Type: Literature]
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3
[SID160673019]
Chemical stability of the compound at pH mimicking gastric juice acidity [AID644883, Type: Literature]
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4
[SID160673019]
Chemical stability of the compound at physiological conditions [AID644884, Type: Literature]
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5
[SID160673019]
EC50 Agonist activity at turkey P2Y purinoceptor 1 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetry [AID647893, Type: Literature]P2Y purinoceptor 1 [gi:1352693]
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6
[SID160673019]
EC50 Agonist activity at human P2Y purinoceptor 2 expressed in human 1321N1 cells assessed as increase in intracellular calcium concentration by spectrofluorimetry [AID647894, Type: Literature]P2Y purinoceptor 2 [gi:311033490]
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7
[SID160673019]
EC50 Activity against human P2Y2-GFP expressed in A549 cells by intracellular calcium increase [AID261699, Type: Literature]P2Y purinoceptor 2 [gi:311033490]
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8
[SID160673019]
EC50 Activity against rat P2Y2-GFP transfected in HEK293 cells by intracellular calcium increase [AID261697, Type: Literature]P2Y purinoceptor 2 [gi:1709518]
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