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sesamol (CID 68289) - Compound BioActivity Data
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BioActivity Outcomes:
Active(14)
 
 
Inactive(221)
 
 
Inconclusive(25)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD PPAR(13)
 
 
 
NR LBD AR(9)
 
 
 
 
NR LBD ER(9)
 
 
 
NR LBD TR(7)
 
 
 
 
NR LBD VDR(6)
 
 
 
BioAssay Types:
Confirmatory(212)
 
 
 
 
Summary(24)
 
 
 
 
Literature(7)
 
 
 
 
Screening(1)
 
 
BioActivity Types:
Potency(194)
 
 
 
 
Kd(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 247    Data Row: 262   Total Pages: 14   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144208409]
Potency-Replicate_1 0.0606qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743040, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
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2
[SID144208409]
Potency-Replicate_1 0.2732qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway [AID743036, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
3
[SID144208409]
Ratio Potency (uM) 0.577411qHTS assay to identify small molecule agonists of the androgen receptor (AR) signaling pathway: Summary [AID743053, Type: summary]AR protein [Homo sapiens] [gi:124375976]
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4
[SID144208409]
Potency-Replicate_1 54.0397qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - wild type cell line [AID743012, Type: confirmatory]
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5
[SID144208409]
Potency-Replicate_1 54.0397qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rev3 mutant cell line [AID743014, Type: confirmatory]
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6
[SID144208409]
TR Potency (uM) 63.0057qHTS assay to identify small molecule antagonists of the thyroid receptor (TR) signaling pathway: Summary [AID743067, Type: summary]thyroid hormone receptor beta isoform 2 [Rattus norvegicus] [gi:399498506]
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7
[SID170482007]
Kd 5500Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Fragment-Based Approach To The Design Of Ligands Targeting A Novel Site In Hiv-1 Integrase [gi:325533893]
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8
[SID170482007]
Kd 5500Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain A, Fragment-Based Approach To The Design Of Ligands Targeting A Novel Site In Hiv-1 Integrase [gi:325533893]
View
9
[SID170482007]
Kd 5500Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain B, Fragment-Based Approach To The Design Of Ligands Targeting A Novel Site In Hiv-1 Integrase [gi:325533894]
View
10
[SID170482007]
Kd 5500Experimentally measured binding affinity data (Kd) for protein-ligand complexes derived from PDB [AID977611, Type: Literature]Chain B, Fragment-Based Approach To The Design Of Ligands Targeting A Novel Site In Hiv-1 Integrase [gi:325533894]
View
11
[SID48414453]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary SingleCellCall Results [AID1189, Type: other]
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12
[SID48414453]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary Mouse Bioassay Results [AID1199, Type: other]
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13
[SID48414453]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary MultiCellCall Results [AID1205, Type: other]
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14
[SID48414453]
DSSTox (CPDBAS) Carcinogenic Potency Database Summary Rat Bioassay Results [AID1208, Type: other]
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15
[SID123096809]
Inhibition of Wnt/beta-catenin signaling pathway in human HEK293 cells at 20 uM after 24 hrs by dual luciferase reporter gene assay relative to vehicle-treated control [AID779150, Type: Literature]
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16
[SID17389735]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838, Type: other]
View
17
[SID144208409]
Potency-Replicate_1 10.7823qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway using the MDA cell line [AID743042, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
View
18
[SID17389735]
Potency 15.8489qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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19
[SID17389735]
Potency qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1 [AID900, Type: confirmatory]caspase-1 isoform alpha precursor [Homo sapiens] [gi:15431328]
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20
[SID11537225]
NMR Based Screening Assay for FKBP12 [AID608, Type: other]peptidyl-prolyl cis-trans isomerase FKBP1A isoform a [Homo sapiens] [gi:17149836]
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