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Prestwick0_001082 (CID 6714004) - Compound BioActivity Data
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BioActivity Outcomes:
Active(10)
 
 
Inactive(62)
 
 
Inconclusive(16)
 
 
Unspecified(3)
 
 
Top Targets:
Pyr redox dim(6)
 
 
 
7TM GPCR Srx(4)
 
 
 
PIKKc TOR(4)
 
 
 
ANK(3)
 
 
PIN FEN1(3)
 
 
BioAssay Types:
Confirmatory(85)
 
 
 
 
 
Literature(5)
 
 
 
Screening(1)
 
 
BioActivity Types:
Potency(86)
 
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 77    Data Row: 91   Total Pages: 5   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID90340893]
Potency 0.0095qHTS Validation Assay for Inhibitors of HP1-beta Chromodomain Interactions with Methylated Histone Tails [AID488953, Type: confirmatory]chromobox protein homolog 1 [Homo sapiens] [gi:187960037]
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2
[SID90340893]
Potency 3.1623qHTS Assay for Identifying Gametocytocidal Compounds [AID743244, Type: confirmatory]
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3
[SID124892371]
Potency 3.9811qHTS for Inhibitors of human tyrosyl-DNA phosphodiesterase 1 (TDP1): qHTS in cells in presence of CPT [AID686979, Type: confirmatory]TDP1 protein [Homo sapiens] [gi:79154014]
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4
[SID50111076]
Potency 7.9433qHTS for inhibitors of binding or entry into cells for Marburg Virus [AID540276, Type: confirmatory]gene 4 small orf - Marburg virus [Marburg marburgvirus] [gi:420597]
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5
[SID90340893]
Potency 8.1961qHTS for Inhibitors of binding or entry into cells for Lassa Virus [AID540256, Type: confirmatory]
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6
[SID90340893]
Potency 9.4662qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory]euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070]
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7
[SID90340893]
Potency 10qHTS for Inhibitors of Glutaminase (GLS): LOPAC Validation [AID624146, Type: confirmatory]GLS protein [Homo sapiens] [gi:71051501]
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8
[SID90340893]
Potency 21.1923Inhibitors of Regulator of G Protein Signaling (RGS) 4: qHTS [AID504845, Type: confirmatory]regulator of G-protein signaling 4 [Homo sapiens] [gi:86301163]
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9
[SID90340893]
Potency 28.1838qHTS for Inhibitors of ATXN expression: Validation of Cytotoxic Assay [AID588349, Type: confirmatory]
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10
[SID90340893]
Potency 28.1838qHTS for Inhibitors of ATXN expression [AID651635, Type: confirmatory]ataxin-2 [Homo sapiens] [gi:171543895]
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11
[SID103279224]
Anticholinesterase activity against erythrocyte acetylcholinesterase (AChE) in humans.(no detectable activity at 3*10e-5 M) [AID31016, Type: Literature]
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12
[SID103279224]
Anticholinesterase activity against plasma Butyrylcholinesterase (BChE) in humans.(no detectable activity at 3*10e-5 M) [AID44276, Type: Literature]
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13
[SID124892371]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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14
[SID90340893]
Potency 0.5623qHTS assay for inhibitors of recombinant human GCK-GKRP interaction: Diaphorase-coupled assay [AID743205, Type: confirmatory]glucokinase regulatory protein [Homo sapiens] [gi:221625433]
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15
[SID90340893]
Potency 0.5623qHTS assay for inhibitors of recombinant human GCK-GKRP interaction: Diaphorase-coupled assay [AID743205, Type: confirmatory]glucokinase isoform 1 [Homo sapiens] [gi:4503951]
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16
[SID124892371]
Potency 12.5893qHTS for Inhibitors of TGF-b: Cytotox Counterscreen [AID588856, Type: confirmatory]
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17
[SID90340893]
Potency 14.6892qHTS for Inducers of the Endoplasmic Reticulum Stress Response (ERSR) in Human Glioma: qHTS [AID602332, Type: confirmatory]heat shock 70kDa protein 5 (glucose-regulated protein, 78kDa) [Homo sapiens] [gi:168984549]
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18
[SID90340893]
Potency 23.1093qHTS for Activators of Parkin Expression: LOPAC Validation Assay (FLuc Reporter) [AID720573, Type: confirmatory]Parkin [Homo sapiens] [gi:3063388]
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19
[SID124892371]
Potency A Quantitative High throughput Screen to Identify Chemical Modulators of PINK1 Expression [AID624263, Type: confirmatory]Parkin [Homo sapiens] [gi:3063388]
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20
[SID90340893]
Potency qHTS for Inhibitors of Polymerase Kappa [AID588579, Type: confirmatory]DNA polymerase kappa [Homo sapiens] [gi:7705344]
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