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BioActivity Data for Compound NCGC00015899-01 (CID 6603988)

BioActivity Outcomes:
Active(6)
 
 
Inactive(62)
 
 
Inconclusive(11)
 
 
Unspecified(1)
 
 
Top Targets:
p450(9)
 
 
 
 
Pyruvate Kina..(4)
 
 
HSD10-like SD..(4)
 
 
GH27(3)
 
 
ampC(2)
 
 
BioAssay Types:
Confirmatory(67)
 
 
 
 
BioAssay Categories:
Toxicity(2)
 
 
BioActivity Types:
Potency(45)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 72    Data Row: 80   Total Pages: 4   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID11111748]
Potency 1qHTS Assay for Inhibitors and Substrates of Cytochrome P450 2D6 [AID891, Type: confirmatory]cytochrome P450 2D6 isoform 1 [Homo sapiens] [gi:40805836]
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2
[SID11111748]
Potency 5.6234qHTS Assay for Antagonists of Acetylcholine Muscarinic M1 Receptor: Kinetic Measurement of Intracellular Calcium Response [AID943, Type: confirmatory]muscarinic acetylcholine receptor M1 [Rattus norvegicus] [gi:18249941]
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3
[SID11111748]
Potency 7.0795qHTS Assay for Antagonists of Acetylcholine Muscarinic M1 Receptor: Measurement of IP-One Response [AID944, Type: confirmatory]muscarinic acetylcholine receptor M1 [Rattus norvegicus] [gi:18249941]
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4
[SID11111748]
Potency 10qHTS Assay for Activators of Cytochrome P450 3A4 [AID885, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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5
[SID11111748]
Cytochrome panel assay with activity outcomes [AID1851_2, Type: other]cytochrome P450 2D6 isoform 2 [Homo sapiens] [gi:68509921]
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6
[SID11111748]
p450-cyp1a2 [AID410, Type: confirmatory]cytochrome P450 1A2 [Homo sapiens] [gi:73915100]
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7
[SID11111748]
Cytochrome panel assay with activity outcomes [AID1851, Type: other]
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8
[SID11111748]
Potency 10qHTS Assay for Inhibitors and Substrates of Cytochrome P450 3A4 [AID884, Type: confirmatory]cytochrome P450 3A4 isoform 1 [Homo sapiens] [gi:13435386]
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9
[SID11111748]
AP1 Signaling Pathway [AID357, Type: confirmatory]
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10
[SID11111748]
Potency qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1: Spectroscopic Profiling in AFC Spectral Region [AID923, Type: confirmatory]
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11
[SID11111748]
Ubiquitin-GFP Assay [AID526, Type: confirmatory]
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12
[SID11111748]
Stat Signaling Pathway [AID446, Type: confirmatory]
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13
[SID11111748]
Potency qHTS Assay for Anthrax Lethal Toxin Internalization [AID912, Type: confirmatory]lethal factor [Bacillus anthracis str. A2012] [gi:21392848]
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14
[SID11111748]
Potency qHTS Assay for Activators of Human Muscle Pyruvate Kinase [AID954, Type: confirmatory]pyruvate kinase PKM isoform b [Homo sapiens] [gi:33286420]
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15
[SID11111748]
Potency qHTS Assay for Inhibitors of Human Muscle Pyruvate Kinase [AID958, Type: confirmatory]pyruvate kinase PKM isoform b [Homo sapiens] [gi:33286420]
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16
[SID11111748]
Potency qHTS Assay for Inhibitors of RGS12 GoLoco Motif Activity (Green Fluorophore) [AID879, Type: confirmatory]guanine nucleotide-binding protein G(i) subunit alpha-1 isoform 1 [Homo sapiens] [gi:33946324]
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17
[SID11111748]
Potency qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor: Activators of Intracellular cAMP Concentrations in Parental HEK 293 [AID938, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
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18
[SID11111748]
Potency qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor [AID926, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
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19
[SID11111748]
Potency qHTS Assay for Inhibitors of Firefly Luciferase [AID411, Type: confirmatory]Luciferase [Photinus pyralis] [gi:160794]
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20
[SID11111748]
Potency Counterscreen for Glucocerebrosidase Inhibitors: qHTS Assay for Human alpha-Galactosidase at pH 4.5 [AID992, Type: confirmatory]alpha-galactosidase [Homo sapiens] [gi:757912]
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