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6-azacytidine (CID 65114) - Compound BioActivity Data
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BioActivity Outcomes:
Active(12)
 
 
Inactive(203)
 
 
Inconclusive(33)
 
 
Unspecified(1)
 
 
Top Targets:
NR LBD PPAR(13)
 
 
 
NR LBD ER(9)
 
 
 
NR LBD AR(9)
 
 
 
 
NR LBD TR(7)
 
 
 
NR LBD VDR(6)
 
 
BioAssay Types:
Confirmatory(213)
 
 
 
 
Summary(24)
 
 
 
 
Literature(1)
 
 
BioActivity Types:
Potency(194)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 238    Data Row: 249   Total Pages: 5   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID17390032]
Potency 0.7943qHTS assay for small molecule activators of the p53 signaling pathway [AID651743, Type: confirmatory]Cellular tumor antigen p53 [gi:269849759]
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2
[SID144208429]
Potency-Replicate_1 1.9351qHTS assay for small molecule agonists of the p53 signaling pathway [AID651631, Type: confirmatory]Cellular tumor antigen p53 [gi:269849759]
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3
[SID144208429]
Ratio Potency (uM) 2.1712qHTS assay for small molecule agonists of the p53 signaling pathway: Summary [AID720552, Type: summary]Cellular tumor antigen p53 [gi:269849759]
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4
[SID17390032]
Potency 5.308qHTS assay for small molecule antagonists of the retinoid-related orphan receptor gamma (ROR-gamma) signaling pathway [AID651802, Type: confirmatory]Nuclear receptor ROR-gamma [gi:49066040]
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5
[SID144208429]
Potency-Replicate_1 6.1193qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - Rad54/Ku70 mutant cell line [AID743015, Type: confirmatory]
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6
[SID144208429]
Potency-Replicate_1 13.6993qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against isogenic chicken DT40 cell lines with known DNA damage response pathways - wild type cell line [AID743012, Type: confirmatory]
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7
[SID17390032]
Potency 22.3872qHTS Assay for Enhancers of SMN2 Splice Variant Expression [AID1458, Type: confirmatory]survival motor neuron protein isoform d [Homo sapiens] [gi:10937869]
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8
[SID17390032]
Potency 25.1189qHTS assay for small molecule antagonists of farnesoid X receptor signaling [AID588526, Type: confirmatory]farnesoid X nuclear receptor [Homo sapiens] [gi:325495553]
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9
[SID144208429]
Potency-Replicate_1 27.5627qHTS assay to identify small molecule antagonists of the farnesoid-X-receptor (FXR) signaling pathway [AID743217, Type: confirmatory]farnesoid X nuclear receptor [Homo sapiens] [gi:325495553]
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10
[SID144208429]
Potency-Replicate_1 30.9258qHTS assay to identify small molecule antagonists of the androgen receptor (AR) signaling pathway [AID743035, Type: confirmatory]AR protein [Homo sapiens] [gi:124375976]
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11
[SID17390032]
Potency 74.978qHTS assay to identify small molecules that stimulate interleukin-8 (IL-8) secretion [AID651758, Type: confirmatory]interleukin 8 [Homo sapiens] [gi:186368]
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12
[SID144208429]
qHTS assay to identify small molecule antagonists of the farnesoid-X-receptor (FXR) signaling pathway: Summary [AID743240, Type: summary]farnesoid X nuclear receptor [Homo sapiens] [gi:325495553]
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13
[SID17390032]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838, Type: other]
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14
[SID17390032]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838_1, Type: other]
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15
[SID17390032]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838_5, Type: other]
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16
[SID17390032]
Potency Cell Viability - LYMP2-004 [AID966, Type: confirmatory]
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17
[SID17390032]
Potency qHTS Assay for Allosteric/Competitive Inhibitors of Caspase-1: Spectroscopic Profiling in AFC Spectral Region [AID923, Type: confirmatory]
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18
[SID17390032]
Potency MultiTox-Fluor Cytotoxicity Assay - LYMP1-001 - Dead Cells [AID946, Type: confirmatory]
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19
[SID17390032]
Potency MultiTox-Fluor Cytotoxicity Assay - LYMP1-001 - Live Cells [AID947, Type: confirmatory]
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20
[SID17390032]
Potency Cell Viability - LYMP1-002 - Assay at 16 hr [AID948, Type: confirmatory]
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21
[SID17390032]
Potency MultiTox-Fluor Cytotoxicity Assay - LYMP1-002 - Live Cells [AID955, Type: confirmatory]
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22
[SID17390032]
Potency MultiTox-Fluor Cytotoxicity Assay - LYMP1-002 - Dead Cells [AID960, Type: confirmatory]
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23
[SID17390032]
Cellular Toxicity (caspase-3) H-4-II-E [AID663, Type: confirmatory]
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24
[SID17390032]
Cellular Toxicity (caspase-3) Hek293 [AID664, Type: confirmatory]
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25
[SID17390032]
Cellular Toxicity (caspase-3) N2a [AID665, Type: confirmatory]
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26
[SID17390032]
Cellular Toxicity (caspase-3) NIH 3T3 [AID666, Type: confirmatory]
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27
[SID17390032]
Cellular Toxicity (caspase-3) Renal Proximal Tubule [AID667, Type: confirmatory]
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28
[SID17390032]
Potency Cell Viability - LYMP2-001 [AID921, Type: confirmatory]
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29
[SID17390032]
Cellular Toxicity (caspase-3) SHSY5Y [AID657, Type: confirmatory]
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30
[SID17390032]
Cellular Toxicity (caspase-3) BJ [AID658, Type: confirmatory]
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31
[SID17390032]
Cellular Toxicity (caspase-3) MRC-5 [AID659, Type: confirmatory]
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32
[SID17390032]
Cellular Toxicity (caspase-3) Mesangial [AID660, Type: confirmatory]
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33
[SID17390032]
Cellular Toxicity (caspase-3) SK-N-SH [AID661, Type: confirmatory]
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34
[SID17390032]
Cell signaling CRE-BLA (Fsk stim) [AID662, Type: confirmatory]
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35
[SID17390032]
Cell Viability - Mesenchymal [AID546, Type: confirmatory]
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36
[SID17390032]
qHTS Assay for Disrupters of an Hsp90 Co-Chaperone Interaction [AID595, Type: confirmatory]
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37
[SID17390032]
qHTS Assay for Inhibitors of DNA Polymerase III Holoenzyme System [AID603, Type: confirmatory]
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38
[SID17390032]
Cellular Toxicity (caspase-3) HepG2 [AID654, Type: confirmatory]
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39
[SID17390032]
Cellular Toxicity (caspase-3) Jurkat [AID655, Type: confirmatory]
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40
[SID17390032]
Cellular Toxicity (caspase-3) HUV-EC-C [AID656, Type: confirmatory]
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41
[SID17390032]
Cell Viability - N2a [AID540, Type: confirmatory]
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42
[SID17390032]
Cell Viability - NIH 3T3 [AID541, Type: confirmatory]
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43
[SID17390032]
Cell Viability - HUV-EC-C [AID542, Type: confirmatory]
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44
[SID17390032]
Cell Viability - H-4-II-E [AID543, Type: confirmatory]
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45
[SID17390032]
Cell Viability - SH-SY5Y [AID544, Type: confirmatory]
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46
[SID17390032]
Cell Viability - Renal Proximal Tubule [AID545, Type: confirmatory]
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47
[SID17390032]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838_4, Type: other]
View
48
[SID17390032]
Potency Cell Viability - LYMP1-002 - Assay at 40 hr [AID994, Type: confirmatory]
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49
[SID17390032]
Potency qHTS Assay for Compounds Blocking the Interaction Between CBF-beta and RUNX1 for the Treatment of Acute Myeloid Leukemia [AID1477, Type: confirmatory]
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50
[SID17390032]
Potency qHTS Assay for Compounds that Induce Erasure of Genomic Imprints [AID1948, Type: confirmatory]
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