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Diacetyl (CID 650) - Compound BioActivity Data
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BioActivity Outcomes:
Active(1)
 
 
Inactive(448)
 
 
Inconclusive(19)
 
 
Unspecified(13)
 
 
Top Targets:
NR LBD PPAR(13)
 
 
 
NR LBD ER(10)
 
 
NR LBD TR(9)
 
 
Esterase lipa..(9)
 
 
NR LBD AR(9)
 
 
BioAssay Types:
Confirmatory(404)
 
 
 
 
Summary(25)
 
 
Literature(18)
 
 
 
Screening(13)
 
 
BioActivity Types:
Potency(364)
 
 
 
 
Ki(10)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 414    Data Row: 481   Total Pages: 25   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID48414775]
DSSTox (DBPCAN) EPA Water Disinfection By-Products with Carcinogenicity Estimates [AID1201, Type: other]
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2
[SID11111061]
Potency 31.6228qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor [AID926, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
View
3
[SID103462449]
Ki 100Inhibition constant against human intestinal carboxylesterase 2 (hiCE) using nitrophenyl acetate (o-NPA) as substrate [AID239272, Type: Literature]Cocaine esterase [gi:46576349]
View
4
[SID103462449]
Ki 100Inhibition of human intestinal carboxylesterase using o-nitrophenyl acetate as substrate after 5 mins by spectrophotometry [AID612131, Type: Literature]Cocaine esterase [gi:46576349]
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5
[SID103462449]
Ki 100Inhibition of rabbit liver carboxylesterase using o-nitrophenyl acetate as substrate after for 5 mins by spectrophotometry [AID612132, Type: Literature]Liver carboxylesterase 1 [gi:51338757]
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6
[SID103462449]
Ki 100Inhibition constant against rabbit liver carboxylesterase (rCE) using nitrophenyl acetate (o-NPA) as substrate [AID239167, Type: Literature]
View
7
[SID103462449]
Ki 100Inhibition of human acetylcholinesterase using acetylthiocholine as substrate by spectrophotometry [AID612134, Type: Literature]Acetylcholinesterase [gi:113037]
View
8
[SID103462449]
Ki 100Inhibition constant against human Acetylcholinesterase (hAcChE) using acetylthiocholine (AcTCh) as substrate [AID239122, Type: Literature]Acetylcholinesterase [gi:113037]
View
9
[SID103462449]
Ki 100Inhibition constant against human Butyrylcholinesterase (hBuChE) using butyrylthiocholine (BuTCh) as substrate [AID239166, Type: Literature]Cholinesterase [gi:116353]
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10
[SID103462449]
Ki 100Inhibition of human butyrylcholinesterase using butyrylthiocholine as substrate by spectrophotometry [AID612135, Type: Literature]Cholinesterase [gi:116353]
View
11
[SID103462449]
Ki 100Inhibition of human liver carboxylesterase1 using o-nitrophenyl acetate as substrate after 5 mins by spectrophotometry [AID612130, Type: Literature]Liver carboxylesterase 1 [gi:119576]
View
12
[SID103462449]
Ki 100Inhibition constant against human liver carboxylesterase 1 (hCE1) using nitrophenyl acetate (o-NPA) as substrate [AID239197, Type: Literature]Liver carboxylesterase 1 [gi:119576]
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13
[SID17389666]
qHTS assay for identifying genotoxic compounds that show differential cytotoxicity against a panel of isogenic chicken DT40 cell lines with known DNA damage response pathways [AID651838, Type: other]
View
14
[SID50105421]
Potency qHTS Assay for Inhibitors of MBNL1-poly(CUG) RNA binding [AID2675, Type: confirmatory]muscleblind-like protein 1 isoform a [Homo sapiens] [gi:41281591]
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15
[SID90340673]
Potency 0.151qHTS screen for enhancers of Arylsulfatase A (ASA1): LOPAC Validation Assay [AID720538, Type: confirmatory]arylsulfatase A [Homo sapiens] [gi:220983390]
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16
[SID90340673]
Potency 0.631qHTS for Inhibitors of Glutaminase (GLS): LOPAC Validation [AID624146, Type: confirmatory]GLS protein [Homo sapiens] [gi:71051501]
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17
[SID17389666]
Potency 3.9811qHTS Assay for Agonists of the Thyroid Stimulating Hormone Receptor: Activators of Intracellular cAMP Concentrations in Parental HEK 293 [AID938, Type: confirmatory]thyroid stimulating hormone receptor [Homo sapiens] [gi:38016895]
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18
[SID50105421]
Potency 10qHTS Assay for Inhibitors of Histone Lysine Methyltransferase G9a [AID504332, Type: confirmatory]euchromatic histone-lysine N-methyltransferase 2 [Homo sapiens] [gi:168985070]
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19
[SID90340673]
Potency 44.6684qHTS Validation Assay for Inhibitors of HP1-beta Chromodomain Interactions with Methylated Histone Tails [AID488953, Type: confirmatory]chromobox protein homolog 1 [Homo sapiens] [gi:187960037]
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20
[SID90340673]
Potency qHTS Validation Assay for Inhibitors of Ubiquitin-specific Protease USP2a Using CHOP2 as the Reporter [AID463106, Type: confirmatory]ubiquitin carboxyl-terminal hydrolase 2 isoform a [Homo sapiens] [gi:188528692]
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