Bookmark and Share
1,3-dipropyl-8-(3-noradamantyl)xanthine (CID 64627) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(25)
 
 
Unspecified(61)
 
 
Top Targets:
7tm 4(20)
 
 
 
MFS(4)
 
 
BioAssay Types:
Literature(85)
 
 
 
BioActivity Types:
Ki(23)
 
 
 
IC50(4)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 80    Data Row: 86   Total Pages: 5   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103234175]
Ki 0.000145Binding affinity to mouse adenosine A1 receptor [AID462308, Type: Literature]Adenosine receptor A1 [gi:341940620]
View
2
[SID103234175]
Ki 0.00019Binding affinity towards adenosine A1 receptor in rat forebrain membranes using N6-[3H]cyclohexyladenosine [AID32193, Type: Literature]Adenosine receptor A1 [gi:2827766]
View
3
[SID103234175]
Ki 0.00019Binding affinity at bovine Adenosine A1 receptor. [AID31984, Type: Literature]
View
4
[SID103234175]
Ki 0.000295Binding affinity to human adenosine A1 receptor [AID462302, Type: Literature]Adenosine receptor A1 [gi:231473]
View
5
[SID103234175]
Ki 0.00072Inhibition of binding to membranes from HEK293 cells expressing human Adenosine A1 receptor [AID30772, Type: Literature]Adenosine receptor A1 [gi:231473]
View
6
[SID103234175]
Ki 0.0011Binding affinity for Adenosine A1 receptor from Guinea pig membranes [AID32168, Type: Literature]Adenosine receptor A1 [gi:1351830]
View
7
[SID103234175]
Ki 0.0013Binding affinity towards adenosine A1 receptor using N6-[3H]cyclohexyladenosine in guinea pig forebrain membranes [AID32289, Type: Literature]Adenosine receptor A1 [gi:1351830]
View
8
[SID103234175]
Ki 0.0013Binding affinity against adenosine A1 receptor in guinea pig forebrain membranes using N6-[3H]cyclohexyladenosine as radioligand [AID32292, Type: Literature]Adenosine receptor A1 [gi:1351830]
View
9
[SID103234175]
Ki 0.0013Binding affinity against adenosine A1 receptor using N6-[3H]cyclohexyladenosine as radioligand in guinea pig forebrain membranes [AID32163, Type: Literature]Adenosine receptor A1 [gi:1351830]
View
10
[SID103234175]
Ki 0.0013Binding affinity against adenosine A1 receptor using [3H]-CHA or [3H]PIA as radioligand [AID32177, Type: Literature]
View
11
[SID103234175]
Ki 0.0126Binding affinity for Adenosine A1 receptor of rat forebrain [AID32033, Type: Literature]Adenosine receptor A1 [gi:2827766]
View
12
[SID103234175]
Ki 0.108Inhibition of binding to membranes from HEK293 cells expressing human Adenosine A2 receptor [AID30790, Type: Literature]Adenosine receptor A2a [gi:543740]
View
13
[SID103234175]
Ki 0.108Inhibition of binding to membranes from HEK293 cells expressing human Adenosine A2 receptor [AID30790, Type: Literature]Adenosine receptor A2b [gi:112938]
View
14
[SID103234175]
Ki 0.23Binding affinity for Adenosine A2 receptor from Guinea pig membranes [AID30625, Type: Literature]
View
15
[SID103234175]
Ki 0.38Binding affinity against adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide as radioligand in rat striatal membranes. [AID33563, Type: Literature]
View
16
[SID103234175]
Ki 0.38Binding affinity against adenosine A2 receptor in rat striatal membranes using N-[3H]-ethyladenosin-5''-uronamide as radioligand in the presence of 50 nM cyclopentyladenosine [AID33587, Type: Literature]
View
17
[SID103234175]
Ki 0.43Binding affinity for adenosine A2 receptor using N-[3H]-ethyladenosin-5''-uronamide in guinea pig forebrain membranes [AID30502, Type: Literature]
View
18
[SID103234175]
Ki 0.51Binding affinity for Adenosine A2 receptor from rat striatal membranes [AID33576, Type: Literature]Adenosine receptor A2b [gi:112939]
View
19
[SID103234175]
Ki 0.51Binding affinity for Adenosine A2 receptor from rat striatal membranes [AID33576, Type: Literature]Adenosine receptor A2a [gi:8928539]
View
20
[SID103234175]
IC50 Binding affinity to rat adenosine A1 receptor [AID462305, Type: Literature]Adenosine receptor A1 [gi:2827766]
View