methylamine
(CID
6329
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Inactive(
2
)
Inconclusive(1)
Unspecified(2)
Top Targets:
SLC5sbd CHT(
1
)
BioAssay Types:
Literature(
5
)
BioActivity Types:
Ki(
1
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 5 Data Row: 5 Total Pages: 1
Sort:
[Click the result table header to sort]
#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
103221660
]
Unspecified
Ki
35075.2
Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosome [AID
494749
, Type: Literature]
High affinity choline transporter 1 [gi:
56404887
]
View
X
Row No.
1
Structure
Substance
SID
103221660
CID
6329
Outcome
Unspecified
Ki
35075.2 [uM]
BioAssay
Inhibition of [3H]choline uptake at choline transporter 1 in mouse brain synaptosome
AID
494749
BioAssay type
Literature
Target
High affinity choline transporter 1 [gi:
56404887
]
PubMed
20637607
Data Table
2
[SID
103221660
]
Unspecified
Partition coefficient (logP) [AID
23443
, Type: Literature]
View
X
Row No.
2
Structure
Substance
SID
103221660
CID
6329
Outcome
Unspecified
BioAssay
Partition coefficient (logP)
AID
23443
BioAssay type
Literature
Target
PubMed
3882967
Data Table
3
[SID
103221660
]
Inactive
In vitro inhibitory concentration against chloroquine-resistant Plasmodium falciparum; Not active [AID
158694
, Type: Literature]
View
X
Row No.
3
Structure
Substance
SID
103221660
CID
6329
Outcome
Inactive
BioAssay
In vitro inhibitory concentration against chloroquine-resistant Plasmodium falciparum; Not active
AID
158694
BioAssay type
Literature
Target
PubMed
15026037
Data Table
4
[SID
103221660
]
Inactive
In vitro inhibitory concentration against chloroquine-sensitive Plasmodium falciparum; Not active [AID
158696
, Type: Literature]
View
X
Row No.
4
Structure
Substance
SID
103221660
CID
6329
Outcome
Inactive
BioAssay
In vitro inhibitory concentration against chloroquine-sensitive Plasmodium falciparum; Not active
AID
158696
BioAssay type
Literature
Target
PubMed
15026037
Data Table
5
[SID
103221660
]
Inconclusive
The pKa value was measured at N15 chemical shift changes due to protonation; nd= not determined [AID
233502
, Type: Literature]
View
X
Row No.
5
Structure
Substance
SID
103221660
CID
6329
Outcome
Inconclusive
BioAssay
The pKa value was measured at N15 chemical shift changes due to protonation; nd= not determined
AID
233502
BioAssay type
Literature
Target
PubMed
8246232
Data Table