STK029852 (CID 6322708) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Inactive(2)
 
 
Top Targets:
RGS R7-like(1)
 
 
RGS RGS16(1)
 
 
RGS RGS4(1)
 
 
RGS RGS8(1)
 
 
RGS RZ-like(1)
 
 
BioAssay Types:
Confirmatory(5)
 
 
 
BioActivity Types:
EC50(5)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID57578015]
EC50 0.116Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS16-Galphao for SAR Compounds [AID2298, Type: confirmatory]regulator of G-protein signaling 16 [Homo sapiens] [gi:156416009]
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2
[SID57578015]
EC50 0.123Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS8-Galphao for SAR Compounds [AID2307, Type: confirmatory]RGS8 protein [Homo sapiens] [gi:74355113]
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3
[SID57578015]
EC50 0.164Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds [AID2295, Type: confirmatory]regulator of G-protein signaling 4 [Homo sapiens] [gi:86301151]
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4
[SID57578015]
EC50 0.164Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds [AID2295, Type: confirmatory]regulator of G-protein signaling 4 [Homo sapiens] [gi:86301151]
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5
[SID57578015]
EC50 0.164Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS4-Galphao for SAR compounds [AID2295, Type: confirmatory]regulator of G-protein signaling 4 [Homo sapiens] [gi:86301151]
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6
[SID57578015]
EC50 30Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS7-Galphao for SAR Compounds [AID2296, Type: confirmatory]RGS7 [Homo sapiens] [gi:1166512]
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7
[SID57578015]
EC50 30Dose response, multiplexed high-throughput screen for small molecule regulators of RGS family protein interactions, specifically RGS19-Galphao for SAR Compounds [AID2311, Type: confirmatory]regulator of G-protein signaling 19 [Homo sapiens] [gi:86990435]
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