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carfentanil (CID 62156) - Compound BioActivity Data
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BioActivity Outcomes:
Active(11)
 
 
Unspecified(4)
 
 
Top Targets:
7tm 4(5)
 
 
ERG2 Sigma1R(1)
 
 
BioAssay Types:
Literature(15)
 
 
 
BioActivity Types:
Ki(10)
 
 
EC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 12    Data Row: 15   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103224159]
Ki 2.4e-05Binding affinity against Opioid receptor mu 1 [AID150845, Type: Literature]
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2
[SID103224159]
Ki 9e-05Inhibition of [3H]DAGO binding to rat brain membrane Opioid receptor mu 1 [AID151894, Type: Literature]Mu-type opioid receptor [gi:464314]
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3
[SID103224159]
Ki 0.00025Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family) [AID150398, Type: Literature]Sigma non-opioid intracellular receptor 1 [gi:81882051]
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4
[SID103224159]
Ki 0.00025Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family) [AID150398, Type: Literature]Delta-type opioid receptor [gi:464311]
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5
[SID103224159]
Ki 0.00025Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family) [AID150398, Type: Literature]Kappa-type opioid receptor [gi:464313]
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6
[SID103224159]
Ki 0.00025Inhibition of [3H]diprenorphine binding to rat brain membrane opioid receptors;(T= total opioid receptor family) [AID150398, Type: Literature]Mu-type opioid receptor [gi:464314]
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7
[SID103224159]
EC50 0.0013Inhibition of electrically evoked contraction in guinea pig ileum determined in vitro [AID73902, Type: Literature]
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8
[SID103224159]
Ki 0.00328Binding affinity against Opioid receptor delta 1 [AID150088, Type: Literature]
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9
[SID103224159]
Ki 0.009Opioid receptor kappa 1 apparent binding constant from rat brain membranes using [3H]DADLE binding assay [AID148442, Type: Literature]
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10
[SID103224159]
Ki 0.0431Binding affinity against Opioid receptor kappa 1 [AID148708, Type: Literature]
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11
[SID103224159]
Ki 0.092Opioid receptor kappa 1 apparent binding constant from guinea pig cerebellum using [3H]diprenorphine binding assay [AID149543, Type: Literature]Kappa-type opioid receptor [gi:730228]
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12
[SID103224159]
Duration of analgesic effect calculated using in vivo rat tail withdrawal assay. [AID174621, Type: Literature]
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13
[SID103224159]
Analgesic activity at 1 min following injection at 1 mg/kg into the lateral tail vein of the rat (55 degree Centigrade hot plate assay) [AID177756, Type: Literature]
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14
[SID103224159]
Analgesic effect calculated using in vivo rat tail withdrawal assay. [AID177922, Type: Literature]
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15
[SID103224159]
Binding energy by using the equation deltaG obsd = -RT ln KD [AID227718, Type: Literature]
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