| 1 | [SID103215636] | Active | Km | 21 | Activity of Carnobacterium divergens BM4489 penicillinase Cad-1 assessed as initial rate of hydrolysis by spectrophotometer [AID422496, Type: Literature] | |   View X | Row No. | 1 | | Structure | 
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | Km | 21 [uM] | | BioAssay | Activity of Carnobacterium divergens BM4489 penicillinase Cad-1 assessed as initial rate of hydrolysis by spectrophotometer | | AID | 422496 | | BioAssay type | Literature | | Target | | | PubMed | 18070972 | | Data Table | |
|
| 2 | [SID103215636] | Active | Km | 31 | Activity of Beta-lactamase OXA-1 expressed in Escherichia coli BL21 (DE3) [AID525581, Type: Literature] | | View X | Row No. | 2 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | Km | 31 [uM] | | BioAssay | Activity of Beta-lactamase OXA-1 expressed in Escherichia coli BL21 (DE3) | | AID | 525581 | | BioAssay type | Literature | | Target | | | PubMed | 20086146 | | Data Table | |
|
| 3 | [SID103215636] | Active | Km | 36 | Activity of beta-lactamase FUS1 assessed as compound hydrolysis by spectrophotometry [AID519632, Type: Literature] | | View X | Row No. | 3 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | Km | 36 [uM] | | BioAssay | Activity of beta-lactamase FUS1 assessed as compound hydrolysis by spectrophotometry | | AID | 519632 | | BioAssay type | Literature | | Target | | | PubMed | 18212108 | | Data Table | |
|
| 4 | [SID103215636] | Active | | | Antimicrobial activity against Carnobacterium divergens BM4490 expressing beta-lactamase CAD1 at 3 McFarland inoculum size by E-test [AID422493, Type: Literature] | | View X | Row No. | 4 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antimicrobial activity against Carnobacterium divergens BM4490 expressing beta-lactamase CAD1 at 3 McFarland inoculum size by E-test | | AID | 422493 | | BioAssay type | Literature | | Target | | | PubMed | 18070972 | | Data Table | |
|
| 5 | [SID103215636] | Active | | | Antimicrobial activity against Escherichia coli HN1157/pHSG576oxa7 assessed as minimal drug concentration [AID523272, Type: Literature] | | View X | Row No. | 5 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antimicrobial activity against Escherichia coli HN1157/pHSG576oxa7 assessed as minimal drug concentration | | AID | 523272 | | BioAssay type | Literature | | Target | | | PubMed | 20160052 | | Data Table | |
|
| 6 | [SID103215636] | Active | | | Antimicrobial activity against Carnobacterium divergens BM4490 expressing beta-lactamase CAD1 at 0.5 McFarland inoculum size by E-test [AID425867, Type: Literature] | | View X | Row No. | 6 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antimicrobial activity against Carnobacterium divergens BM4490 expressing beta-lactamase CAD1 at 0.5 McFarland inoculum size by E-test | | AID | 425867 | | BioAssay type | Literature | | Target | | | PubMed | 18070972 | | Data Table | |
|
| 7 | [SID103215636] | Active | | | Induction of Ppbp2::lacZ gene expression in Staphylococcus aureus SH1000 at 0.3 ug/ml after 0.5 hrs by beta-galactosidase reporter gene assay relative to untreated control [AID530763, Type: Literature] | | View X | Row No. | 7 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of Ppbp2::lacZ gene expression in Staphylococcus aureus SH1000 at 0.3 ug/ml after 0.5 hrs by beta-galactosidase reporter gene assay relative to untreated control | | AID | 530763 | | BioAssay type | Literature | | Target | | | PubMed | 18541730 | | Data Table | |
|
| 8 | [SID103215636] | Active | | | Induction of Ppbp2::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control [AID530764, Type: Literature] | | View X | Row No. | 8 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of Ppbp2::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control | | AID | 530764 | | BioAssay type | Literature | | Target | | | PubMed | 18541730 | | Data Table | |
|
| 9 | [SID103215636] | Active | | | Induction of PvraSr::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control [AID530765, Type: Literature] | | View X | Row No. | 9 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of PvraSr::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control | | AID | 530765 | | BioAssay type | Literature | | Target | | | PubMed | 18541730 | | Data Table | |
|
| 10 | [SID103215636] | Active | | | Induction of PtcaA::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control [AID530766, Type: Literature] | | View X | Row No. | 10 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of PtcaA::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control | | AID | 530766 | | BioAssay type | Literature | | Target | | | PubMed | 18541730 | | Data Table | |
|
| 11 | [SID103215636] | Active | | | Induction of PlytR::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control [AID530767, Type: Literature] | | View X | Row No. | 11 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of PlytR::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control | | AID | 530767 | | BioAssay type | Literature | | Target | | | PubMed | 18541730 | | Data Table | |
|
| 12 | [SID103215636] | Active | | | Induction of PsgtB::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control [AID530768, Type: Literature] | | View X | Row No. | 12 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of PsgtB::lacZ gene expression in Staphylococcus aureus SH1000 at 8 ug/ml after 2 hrs by beta-galactosidase reporter gene assay relative to untreated control | | AID | 530768 | | BioAssay type | Literature | | Target | | | PubMed | 18541730 | | Data Table | |
|
| 13 | [SID103215636] | Active | | | Binding affinity to Escherichia coli isolate HN1157 AcrAB-TolC efflux transporter [AID523269, Type: Literature] | | View X | Row No. | 13 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Binding affinity to Escherichia coli isolate HN1157 AcrAB-TolC efflux transporter | | AID | 523269 | | BioAssay type | Literature | | Target | | | PubMed | 20160052 | | Data Table | |
|
| 14 | [SID103215636] | Active | | | Antibacterial activity against Escherichia coli NKE1355 harboring deletion mutation in acrB protein and plasmid expressing BAD gene in presence of increasing concentration of arabinose [AID524394, Type: Literature] | | View X | Row No. | 14 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Escherichia coli NKE1355 harboring deletion mutation in acrB protein and plasmid expressing BAD gene in presence of increasing concentration of arabinose | | AID | 524394 | | BioAssay type | Literature | | Target | | | PubMed | 20211889 | | Data Table | |
|
| 15 | [SID103215636] | Active | | | Displacement of benzyl-[14C]penicillin from Staphylococcus aureus PBP2a RU130 mutant at 2500 ug/ml by in vitro competitive assay [AID529299, Type: Literature] | | View X | Row No. | 15 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Displacement of benzyl-[14C]penicillin from Staphylococcus aureus PBP2a RU130 mutant at 2500 ug/ml by in vitro competitive assay | | AID | 529299 | | BioAssay type | Literature | | Target | | | PubMed | 18505853 | | Data Table | |
|
| 16 | [SID103215636] | Active | | | Antimicrobial activity against Bacillus anthracis MurA1 AS clone 2G2 assessed as growth inhibition in presence of xylose by antisense-induced hypersensitive testing [AID529554, Type: Literature] | | View X | Row No. | 16 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antimicrobial activity against Bacillus anthracis MurA1 AS clone 2G2 assessed as growth inhibition in presence of xylose by antisense-induced hypersensitive testing | | AID | 529554 | | BioAssay type | Literature | | Target | | | PubMed | 18378720 | | Data Table | |
|
| 17 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus isolate 1306 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay [AID544606, Type: Literature] | | View X | Row No. | 17 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus isolate 1306 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay | | AID | 544606 | | BioAssay type | Literature | | Target | | | PubMed | 18694946 | | Data Table | |
|
| 18 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus isolate 1326 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay [AID544607, Type: Literature] | | View X | Row No. | 18 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus isolate 1326 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay | | AID | 544607 | | BioAssay type | Literature | | Target | | | PubMed | 18694946 | | Data Table | |
|
| 19 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus isolate 1552 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay [AID544608, Type: Literature] | | View X | Row No. | 19 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus isolate 1552 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay | | AID | 544608 | | BioAssay type | Literature | | Target | | | PubMed | 18694946 | | Data Table | |
|
| 20 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus isolate 4666 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay [AID544609, Type: Literature] | | View X | Row No. | 20 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus isolate 4666 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay | | AID | 544609 | | BioAssay type | Literature | | Target | | | PubMed | 18694946 | | Data Table | |
|
| 21 | [SID103215636] | Active | | | Antibacterial activity against mecA-negative Staphylococcus aureus isolate 29213 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay [AID544610, Type: Literature] | | View X | Row No. | 21 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against mecA-negative Staphylococcus aureus isolate 29213 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay | | AID | 544610 | | BioAssay type | Literature | | Target | | | PubMed | 18694946 | | Data Table | |
|
| 22 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus isolate 6083 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay [AID544611, Type: Literature] | | View X | Row No. | 22 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus isolate 6083 assessed as reduction in bacterial count at 20 ug/ml after 24 hrs by time-kill assay | | AID | 544611 | | BioAssay type | Literature | | Target | | | PubMed | 18694946 | | Data Table | |
|
| 23 | [SID103215636] | Active | | | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20010734 in CYY medium [AID285358, Type: Literature] | | View X | Row No. | 23 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20010734 in CYY medium | | AID | 285358 | | BioAssay type | Literature | | Target | | | PubMed | 17242137 | | Data Table | |
|
| 24 | [SID103215636] | Active | | | Increase in Panton-Valentine leukocidin level in Staphylococcus aureus LUG855 in CCY medium [AID285359, Type: Literature] | | View X | Row No. | 24 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Increase in Panton-Valentine leukocidin level in Staphylococcus aureus LUG855 in CCY medium | | AID | 285359 | | BioAssay type | Literature | | Target | | | PubMed | 17242137 | | Data Table | |
|
| 25 | [SID103215636] | Active | | | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20030203 in CYY medium [AID285360, Type: Literature] | | View X | Row No. | 25 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20030203 in CYY medium | | AID | 285360 | | BioAssay type | Literature | | Target | | | PubMed | 17242137 | | Data Table | |
|
| 26 | [SID103215636] | Active | | | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20040332 in CYY medium [AID285361, Type: Literature] | | View X | Row No. | 26 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20040332 in CYY medium | | AID | 285361 | | BioAssay type | Literature | | Target | | | PubMed | 17242137 | | Data Table | |
|
| 27 | [SID103215636] | Active | | | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20041010 in CYY medium [AID285362, Type: Literature] | | View X | Row No. | 27 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Increase in Panton-Valentine leukocidin level in community acquired methicillin-resistant Staphylococcus aureus HT20041010 in CYY medium | | AID | 285362 | | BioAssay type | Literature | | Target | | | PubMed | 17242137 | | Data Table | |
|
| 28 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus Mu50 assessed as inhibition of bacterial population at greater than 512 ug/ml after 48 hrs [AID325476, Type: Literature] | | View X | Row No. | 28 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus Mu50 assessed as inhibition of bacterial population at greater than 512 ug/ml after 48 hrs | | AID | 325476 | | BioAssay type | Literature | | Target | | | PubMed | 17438056 | | Data Table | |
|
| 29 | [SID103215636] | Active | | | Induction of VraSR-dependent tcaA gene expression in Staphylococcus aureus N315 at 10 ug/mL after 30 mins by Northern blot analysis [AID373187, Type: Literature] | | View X | Row No. | 29 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of VraSR-dependent tcaA gene expression in Staphylococcus aureus N315 at 10 ug/mL after 30 mins by Northern blot analysis | | AID | 373187 | | BioAssay type | Literature | | Target | | | PubMed | 17709474 | | Data Table | |
|
| 30 | [SID103215636] | Active | | | Induction of VraSR-dependent tcaA gene expression in Staphylococcus aureus N315 at 16 ug/mL after 30 mins by Northern blot analysis [AID373188, Type: Literature] | | View X | Row No. | 30 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of VraSR-dependent tcaA gene expression in Staphylococcus aureus N315 at 16 ug/mL after 30 mins by Northern blot analysis | | AID | 373188 | | BioAssay type | Literature | | Target | | | PubMed | 17709474 | | Data Table | |
|
| 31 | [SID103215636] | Active | | | Induction of blaI mRNA expression in methicillin-resistant Staphylococcus aureus 2884 isolateby RT-PCR [AID405584, Type: Literature] | | View X | Row No. | 31 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of blaI mRNA expression in methicillin-resistant Staphylococcus aureus 2884 isolateby RT-PCR | | AID | 405584 | | BioAssay type | Literature | | Target | | | PubMed | 17470657 | | Data Table | |
|
| 32 | [SID103215636] | Active | | | Decrease in PBP2 gene expression in oxacillin-dependent methicillin-resistant Staphylococcus aureus 2884D isolate by RT-PCR [AID405587, Type: Literature] | | View X | Row No. | 32 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Decrease in PBP2 gene expression in oxacillin-dependent methicillin-resistant Staphylococcus aureus 2884D isolate by RT-PCR | | AID | 405587 | | BioAssay type | Literature | | Target | | | PubMed | 17470657 | | Data Table | |
|
| 33 | [SID103215636] | Active | | | Antibacterial activity against Staphylococcus aureus SCV isolated from cystic fibrosis patient infected in human THP-1 cells assessed as log reduction of intracellular CFU level after 24 hrs in presence of thymidine [AID581667, Type: Literature] | | View X | Row No. | 33 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against Staphylococcus aureus SCV isolated from cystic fibrosis patient infected in human THP-1 cells assessed as log reduction of intracellular CFU level after 24 hrs in presence of thymidine | | AID | 581667 | | BioAssay type | Literature | | Target | | | PubMed | 19188393 | | Data Table | |
|
| 34 | [SID103215636] | Active | | | Antibacterial activity against revertant Staphylococcus aureus infected in human THP-1 cells assessed as log reduction of extracellular CFU level after 24 hrs [AID581668, Type: Literature] | | View X | Row No. | 34 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against revertant Staphylococcus aureus infected in human THP-1 cells assessed as log reduction of extracellular CFU level after 24 hrs | | AID | 581668 | | BioAssay type | Literature | | Target | | | PubMed | 19188393 | | Data Table | |
|
| 35 | [SID103215636] | Active | | | Antibacterial activity against normal phenotype Staphylococcus aureus in infected in human THP-1 cells assessed as log reduction of extracellular CFU level after 24 hrs [AID581669, Type: Literature] | | View X | Row No. | 35 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Antibacterial activity against normal phenotype Staphylococcus aureus in infected in human THP-1 cells assessed as log reduction of extracellular CFU level after 24 hrs | | AID | 581669 | | BioAssay type | Literature | | Target | | | PubMed | 19188393 | | Data Table | |
|
| 36 | [SID103215636] | Active | | | Decrease in delta toxin levels in Staphylococcus aureus USA300 at subinhibitory concentrations after 24 hrs by RP-HPLC/ESI- MS [AID574552, Type: Literature] | | View X | Row No. | 36 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Decrease in delta toxin levels in Staphylococcus aureus USA300 at subinhibitory concentrations after 24 hrs by RP-HPLC/ESI- MS | | AID | 574552 | | BioAssay type | Literature | | Target | | | PubMed | 20713669 | | Data Table | |
|
| 37 | [SID103215636] | Active | | | Decrease in PSMbeta1 levels in Staphylococcus aureus Sanger 252 at subinhibitory concentrations after 24 hrs by RP-HPLC/ESI- MS [AID574553, Type: Literature] | | View X | Row No. | 37 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Decrease in PSMbeta1 levels in Staphylococcus aureus Sanger 252 at subinhibitory concentrations after 24 hrs by RP-HPLC/ESI- MS | | AID | 574553 | | BioAssay type | Literature | | Target | | | PubMed | 20713669 | | Data Table | |
|
| 38 | [SID103215636] | Active | | | Decrease in PSMbeta1 levels in Staphylococcus aureus USA300 at subinhibitory concentration after 24 hrs by RP-HPLC/ESI-MS [AID574554, Type: Literature] | | View X | Row No. | 38 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Decrease in PSMbeta1 levels in Staphylococcus aureus USA300 at subinhibitory concentration after 24 hrs by RP-HPLC/ESI-MS | | AID | 574554 | | BioAssay type | Literature | | Target | | | PubMed | 20713669 | | Data Table | |
|
| 39 | [SID48416356] | Active | | | DSSTox (FDAMDD) FDA Maximum (Recommended) Daily Dose Database [AID1195, Type: other] | | View X | Row No. | 39 | | Structure |
| | Substance | | | SID | 48416356 | | CID | 6196 | | Outcome | Active | | BioAssay | DSSTox (FDAMDD) FDA Maximum (Recommended) Daily Dose Database | | AID | 1195 | | BioAssay type | other | | Target | | | PubMed | | | Data Table | |
|
| 40 | [SID103215636] | Active | | | Induction of blaR1 gene expression in oxacillin-dependent methicillin-resistant Staphylococcus aureus 2884D isolate by RT-PCR [AID405644, Type: Literature] | | View X | Row No. | 40 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Induction of blaR1 gene expression in oxacillin-dependent methicillin-resistant Staphylococcus aureus 2884D isolate by RT-PCR | | AID | 405644 | | BioAssay type | Literature | | Target | | | PubMed | 17470657 | | Data Table | |
|
| 41 | [SID103215636] | Active | | | Decrease in PSMalpha levels in Staphylococcus aureus USA300 at subinhibitory concentration after 24 hrs by RP-HPLC/ESI-MS [AID574549, Type: Literature] | | View X | Row No. | 41 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Active | | BioAssay | Decrease in PSMalpha levels in Staphylococcus aureus USA300 at subinhibitory concentration after 24 hrs by RP-HPLC/ESI-MS | | AID | 574549 | | BioAssay type | Literature | | Target | | | PubMed | 20713669 | | Data Table | |
|
| 42 | [SID103215636] | Unspecified | Km | 52 | Activity at Escherichia coli isolate 7181 beta-lactamase OXA-7 [AID523266, Type: Literature] | | View X | Row No. | 42 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | Km | 52 [uM] | | BioAssay | Activity at Escherichia coli isolate 7181 beta-lactamase OXA-7 | | AID | 523266 | | BioAssay type | Literature | | Target | | | PubMed | 20160052 | | Data Table | |
|
| 43 | [SID103215636] | Unspecified | MIC | 79 | Antibacterial activity against Staphylococcus aureus EMRSA-15 after 24 hrs [AID658537, Type: Literature] | | View X | Row No. | 43 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | MIC | 79 [uM] | | BioAssay | Antibacterial activity against Staphylococcus aureus EMRSA-15 after 24 hrs | | AID | 658537 | | BioAssay type | Literature | | Target | | | PubMed | 21899267 | | Data Table | |
|
| 44 | [SID103215636] | Unspecified | Km | 110 | Activity at Pseudomonas fluorescens PF-1 beta-lactamase BIC-1 expressed in Escherichia coli DH10B carrying pSau1 [AID495797, Type: Literature] | | View X | Row No. | 44 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | Km | 110 [uM] | | BioAssay | Activity at Pseudomonas fluorescens PF-1 beta-lactamase BIC-1 expressed in Escherichia coli DH10B carrying pSau1 | | AID | 495797 | | BioAssay type | Literature | | Target | | | PubMed | 19901091 | | Data Table | |
|
| 45 | [SID103215636] | Unspecified | Km | 115 | Activity of Brachyspira pilosicoli beta-lactamase OXA-63 expressed in Escherichia coli BL21 (DE3) assessed as compound hydrolysis by spectrophotometry [AID519631, Type: Literature] | | View X | Row No. | 45 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | Km | 115 [uM] | | BioAssay | Activity of Brachyspira pilosicoli beta-lactamase OXA-63 expressed in Escherichia coli BL21 (DE3) assessed as compound hydrolysis by spectrophotometry | | AID | 519631 | | BioAssay type | Literature | | Target | | | PubMed | 18212108 | | Data Table | |
|
| 46 | [SID103215636] | Unspecified | Km | 450 | Activity of Escherichia coli TOP10 beta-lactamase OXA-143 [AID564228, Type: Literature] | | View X | Row No. | 46 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | Km | 450 [uM] | | BioAssay | Activity of Escherichia coli TOP10 beta-lactamase OXA-143 | | AID | 564228 | | BioAssay type | Literature | | Target | | | PubMed | 19770279 | | Data Table | |
|
| 47 | [SID103215636] | Unspecified | IC50 | 710 | Inhibition of methicillin-resistant Staphylococcus aureus COL PBP2a by competitive assay [AID529294, Type: Literature] | | View X | Row No. | 47 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | IC50 | 710 [uM] | | BioAssay | Inhibition of methicillin-resistant Staphylococcus aureus COL PBP2a by competitive assay | | AID | 529294 | | BioAssay type | Literature | | Target | | | PubMed | 18505853 | | Data Table | |
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| 48 | [SID103215636] | Unspecified | MIC | 1276 | Antibacterial activity against Staphylococcus aureus EMRSA-16 after 24 hrs [AID658538, Type: Literature] | | View X | Row No. | 48 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | MIC | 1276 [uM] | | BioAssay | Antibacterial activity against Staphylococcus aureus EMRSA-16 after 24 hrs | | AID | 658538 | | BioAssay type | Literature | | Target | | | PubMed | 21899267 | | Data Table | |
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| 49 | [SID103215636] | Unspecified | Ki | 3300 | Binding affinity to human PepT2 in SKTP cells [AID612540, Type: Literature] | Solute carrier family 15 member 2 [gi:209572672] | View X | Row No. | 49 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | Ki | 3300 [uM] | | BioAssay | Binding affinity to human PepT2 in SKTP cells | | AID | 612540 | | BioAssay type | Literature | | Target | Solute carrier family 15 member 2 [gi:209572672] | | PubMed | 21741846 | | Data Table | |
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| 50 | [SID103215636] | Unspecified | Ki | 3300 | TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in SKPT cells [AID681114, Type: other] | Solute carrier family 15 member 2 [gi:2499990] | View X | Row No. | 50 | | Structure |
| | Substance | | | SID | 103215636 | | CID | 6196 | | Outcome | Unspecified | | Ki | 3300 [uM] | | BioAssay | TP_TRANSPORTER: inhibition of Gly-Sar uptake (pH6.0) in SKPT cells | | AID | 681114 | | BioAssay type | other | | Target | Solute carrier family 15 member 2 [gi:2499990] | | PubMed | | | Data Table | |
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Chemical Probe 
Active 
Inactive 
Inconclusive 
Unspecified 
