BRD-K43358885-001-01-4
(CID
60193900
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(
1
)
Inactive(
4
)
Top Targets:
FGF(
1
)
rad52(
1
)
BioAssay Types:
Screening(
5
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 5 Data Row: 5 Total Pages: 1
Sort:
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
144200036
]
Active
DENV2 CPE-Based HTS Measured in Cell-Based and Microorganism Combination System Using Plate Reader - 2149-01_Other_SinglePoint_HTS_Activity [AID
651640
, Type: screening]
View
X
Row No.
1
Structure
Substance
SID
144200036
CID
60193900
Outcome
Active
BioAssay
DENV2 CPE-Based HTS Measured in Cell-Based and Microorganism Combination System Using Plate Reader - 2149-01_Other_SinglePoint_HTS_Activity
AID
651640
BioAssay type
screening
Target
PubMed
Data Table
2
[SID
144200036
]
Inactive
Luminescence Cell-Based Primary HTS to identify inhibitors of the oncoprotein EWS/Fli transcriptional activity Measured in Cell-Based System Using Plate Reader - 7014-01_Inhibitor_SinglePoint_HTS_Activity [AID
651661
, Type: screening]
View
X
Row No.
2
Structure
Substance
SID
144200036
CID
60193900
Outcome
Inactive
BioAssay
Luminescence Cell-Based Primary HTS to identify inhibitors of the oncoprotein EWS/Fli transcriptional activity Measured in Cell-Based System Using Plate Reader - 7014-01_Inhibitor_SinglePoint_HTS_Activity
AID
651661
BioAssay type
screening
Target
PubMed
Data Table
3
[SID
144200036
]
Inactive
HTS for PAX8 inhibitors using PAX8 luciferase reporter gene assay in RMG-I cells Measured in Cell-Based System Using Plate Reader - 7054-01_Inhibitor_SinglePoint_HTS_Activity [AID
652154
, Type: screening]
View
X
Row No.
3
Structure
Substance
SID
144200036
CID
60193900
Outcome
Inactive
BioAssay
HTS for PAX8 inhibitors using PAX8 luciferase reporter gene assay in RMG-I cells Measured in Cell-Based System Using Plate Reader - 7054-01_Inhibitor_SinglePoint_HTS_Activity
AID
652154
BioAssay type
screening
Target
PubMed
Data Table
4
[SID
144200036
]
Inactive
FRET-based HTS for detection of RAD52 Inhibitors Measured in Biochemical System Using Plate Reader - 7018-01_Inhibitor_SinglePoint_HTS_Activity_Set2 [AID
651710
, Type: screening]
RAD52 gene product [Homo sapiens] [gi:
109637798
]
View
X
Row No.
4
Structure
Substance
SID
144200036
CID
60193900
Outcome
Inactive
BioAssay
FRET-based HTS for detection of RAD52 Inhibitors Measured in Biochemical System Using Plate Reader - 7018-01_Inhibitor_SinglePoint_HTS_Activity_Set2
AID
651710
BioAssay type
screening
Target
RAD52 gene product [Homo sapiens] [gi:
109637798
]
PubMed
Data Table
5
[SID
144200036
]
Inactive
Small Molecule Inhibitors of FGF22-Mediated Excitatory Synaptogenesis & Epilepsy Measured in Biochemical System Using RT-PCR - 7012-01_Inhibitor_SinglePoint_HTS_Activity [AID
651658
, Type: screening]
FGF22 gene product [Homo sapiens] [gi:
10190672
]
View
X
Row No.
5
Structure
Substance
SID
144200036
CID
60193900
Outcome
Inactive
BioAssay
Small Molecule Inhibitors of FGF22-Mediated Excitatory Synaptogenesis & Epilepsy Measured in Biochemical System Using RT-PCR - 7012-01_Inhibitor_SinglePoint_HTS_Activity
AID
651658
BioAssay type
screening
Target
FGF22 gene product [Homo sapiens] [gi:
10190672
]
PubMed
Data Table