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BRD-K36125895-004-01-8 (CID 60190920) - Compound BioActivity Data
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BioActivity Outcomes:
Active(11)
 
 
Inactive(28)
 
 
Inconclusive(4)
 
 
Top Targets:
PAX(8)
 
 
 
 
rad52(1)
 
 
M1 APN 2(1)
 
 
S-100(1)
 
 
CLECT selecti..(1)
 
 
BioAssay Types:
Screening(23)
 
 
 
Confirmatory(20)
 
 
 
 
BioActivity Types:
AC50(20)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 43    Data Row: 43   Total Pages: 3   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID144196939]
AC50_uM 0.00447SA7-Pax8: cytotoxicity COV434 Measured in Cell-Based System Using Plate Reader - 7054-09_Inhibitor_Dose_DryPowder_Activity [AID743145, Type: confirmatory]PAX8 [Homo sapiens] [gi:998701]
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2
[SID144196939]
AC50_uM 3.15HTS for PAX8 inhibitors using PAX8 luciferase reporter gene assay in RMG-I cells Measured in Cell-Based System Using Plate Reader - 7054-01_Inhibitor_Dose_CherryPick_Activity [AID687027, Type: confirmatory]PAX8 [Homo sapiens] [gi:998701]
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3
[SID144196939]
AC50_uM 5.77PAX8: PAX8-dependent cytoxicity Measured in Cell-Based System Using Plate Reader - 7054-06_Inhibitor_Dose_DryPowder_Activity [AID743049, Type: confirmatory]
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4
[SID144196939]
AC50_uM 17.03Cell fusion assay for clade C HIV-1ZM109 Env Measured in Cell-Based System Using Plate Reader - 7013-05_Inhibitor_Dose_CherryPick_Activity [AID652058, Type: confirmatory]
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5
[SID144196939]
AC50_uM 17.78HIV entry: Env-mediated Cell Fusion Measured in Cell-Based System Using Plate Reader - 7013-01_Inhibitor_Dose_CherryPick_Activity [AID652057, Type: confirmatory]
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6
[SID144196939]
AC50_uM 20.02HIV-1 Cell Fusion assay for clade B Env AD8 Measured in Cell-Based System Using Plate Reader - 7013-04_Inhibitor_Dose_CherryPick_Activity [AID652062, Type: confirmatory]
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7
[SID144196939]
AC50_uM 30.11SA2 PAX8:selectivity PAX5 Measured in Cell-Based System Using Plate Reader - 7054-03_Inhibitor_Dose_DryPowder_Activity [AID743047, Type: confirmatory]
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8
[SID144196939]
AC50_uM 30.84Pax8 Selectivity: PAx2 Measured in Cell-Based System Using Plate Reader - 7054-02_Inhibitor_Dose_DryPowder_Activity [AID743048, Type: confirmatory]
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9
[SID144196939]
AC50_uM 37.88SA11 PAX8: cytotoxicity OVCAR4 Measured in Cell-Based System Using Plate Reader - 7054-13_Inhibitor_Dose_DryPowder_Activity [AID743150, Type: confirmatory]PAX8 [Homo sapiens] [gi:998701]
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10
[SID144196939]
HIV entry: Env-mediated Cell Fusion Measured in Cell-Based System Using Plate Reader - 7013-01_Inhibitor_SinglePoint_HTS_Activity [AID651610, Type: screening]
View
11
[SID144196939]
HTS for PAX8 inhibitors using PAX8 luciferase reporter gene assay in RMG-I cells Measured in Cell-Based System Using Plate Reader - 7054-01_Inhibitor_SinglePoint_HTS_Activity [AID652154, Type: screening]PAX8 [Homo sapiens] [gi:998701]
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12
[SID144196939]
AC50_uM SA8-Pax8: cytotoxicity OV-90 Measured in Cell-Based System Using Plate Reader - 7054-10_Inhibitor_Dose_DryPowder_Activity [AID743149, Type: confirmatory]PAX8 [Homo sapiens] [gi:998701]
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13
[SID144196939]
DENV2 CPE-Based HTS Measured in Cell-Based and Microorganism Combination System Using Plate Reader - 2149-01_Other_SinglePoint_HTS_Activity [AID651640, Type: screening]
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14
[SID144196939]
Luminescence Cell-Based Primary HTS to identify inhibitors of the oncoprotein EWS/Fli transcriptional activity Measured in Cell-Based System Using Plate Reader - 7014-01_Inhibitor_SinglePoint_HTS_Activity [AID651661, Type: screening]
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15
[SID144196939]
MLPCN PGC1a Modulators Measured in Cell-Based System Using Plate Reader - 2139-01_Inhibitor_SinglePoint_HTS_Activity [AID651687, Type: screening]
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16
[SID144196939]
MLPCN PGC1a Modulators Measured in Cell-Based System Using Plate Reader - 2139-01_Activator_SinglePoint_HTS_Activity [AID651723, Type: screening]
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17
[SID144196939]
AC50_uM SA6-Pax8: cytotoxicity A2780 Measured in Cell-Based System Using Plate Reader - 7054-08_Inhibitor_Dose_DryPowder_Activity [AID743046, Type: confirmatory]
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18
[SID144196939]
7011-01_Antagonist_SinglePoint_HTS_Activity [AID720647, Type: screening]
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19
[SID144196939]
HTS for Bacterial rRNA inhibitors Measured in Microorganism-Based System Using Plate Reader - 7056-01_Inhibitor_SinglePoint_HTS_Activity [AID720706, Type: screening]
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20
[SID144196939]
AC50_uM Counterscreen:CMV reporter Measured in Cell-Based System Using Plate Reader - 7054-04_Inhibitor_Dose_DryPowder_Activity [AID743020, Type: confirmatory]
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