AC1NZ8OG (CID 5927555) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(9)
 
 
Inactive(738)
 
 
Inconclusive(12)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srx(20)
 
 
alkPPc(14)
 
 
Bcl-2 like(11)
 
 
Tryp SPc(10)
 
 
 
7TM GPCR Srsx(10)
 
 
BioAssay Types:
Screening(521)
 
 
 
 
 
Confirmatory(222)
 
 
 
 
 
Literature(5)
 
 
BioActivity Types:
Potency(147)
 
 
 
 
IC50(43)
 
 
EC50(10)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 761    Data Row: 761   Total Pages: 16   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID7973802]
 A qHTS for Small Molecule Inhibitors of Shiga Toxin [AID2315, Type: screening]shiga toxin 1 variant A subunit [Escherichia coli O157:H7] [gi:32400299]
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2
[SID7973802]
 Luminescence-based cell-based high throughput confirmation assay for activators of the Aryl Hydrocarbon Receptor (AHR) [AID2845, Type: screening]aryl hydrocarbon receptor precursor [Homo sapiens] [gi:4502003]
View
3
[SID7973802]
 Luminescence-based cell-based high throughput confirmation assay for activators of the Aryl Hydrocarbon Receptor (AHR) [AID2845, Type: screening]aryl hydrocarbon receptor precursor [Homo sapiens] [gi:4502003]
View
4
[SID7973802]
 Luminescence-based cell-based high throughput confirmation assay for activators of the Aryl Hydrocarbon Receptor (AHR) [AID2845, Type: screening]aryl hydrocarbon receptor precursor [Homo sapiens] [gi:4502003]
View
5
[SID7973802]
 Luminescence-based primary cell-based high throughput screening assay to identify activators of the Aryl Hydrocarbon Receptor (AHR) [AID2796, Type: screening]aryl hydrocarbon receptor precursor [Homo sapiens] [gi:4502003]
View
6
[SID7973802]
 Luminescence-based primary cell-based high throughput screening assay to identify activators of the Aryl Hydrocarbon Receptor (AHR) [AID2796, Type: screening]aryl hydrocarbon receptor precursor [Homo sapiens] [gi:4502003]
View
7
[SID7973802]
 Luminescence-based primary cell-based high throughput screening assay to identify activators of the Aryl Hydrocarbon Receptor (AHR) [AID2796, Type: screening]aryl hydrocarbon receptor precursor [Homo sapiens] [gi:4502003]
View
8
[SID7973802]
 Counterscreen for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA): A cell-based dose-response assay for inhibition of the Steroidogenic Factor 1 (SF-1) [AID695, Type: confirmatory]NR5A1 gene product [Homo sapiens] [gi:20070193]
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9
[SID7973802]
 Counterscreen for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA): A cell-based dose-response assay for inhibition of the Steroidogenic Factor 1 (SF-1) [AID695, Type: confirmatory]NR5A1 gene product [Homo sapiens] [gi:20070193]
View
10
[SID7973802]
 Counterscreen for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA): A cell-based dose-response assay for inhibition of the Steroidogenic Factor 1 (SF-1) [AID695, Type: confirmatory]NR5A1 gene product [Homo sapiens] [gi:20070193]
View
11
[SID7973802]
 MLPCN Alpha-Synuclein 5'UTR - 5'-UTR binding - activators [AID1814, Type: screening]
View
12
[SID7973802]
 Counterscreen for activators of the Aryl Hydrocarbon Receptor (AHR): luminescence-based cell-based high throughput screening assay to identify activators of the Pregnane X Receptor (PXR) [AID434939, Type: screening]nuclear receptor subfamily 1 group I member 2 isoform 1 [Homo sapiens] [gi:34398348]
View
13
[SID7973802]
 Counterscreen for activators of the Aryl Hydrocarbon Receptor (AHR): luminescence-based cell-based high throughput screening assay to identify activators of the Pregnane X Receptor (PXR) [AID434939, Type: screening]nuclear receptor subfamily 1 group I member 2 isoform 1 [Homo sapiens] [gi:34398348]
View
14
[SID7973802]
 Kallikrein 5 1536 HTS [AID873, Type: screening]kallikrein-related peptidase 5 preproprotein [Homo sapiens] [gi:6912644]
View
15
[SID7973802]
 Kallikrein 5 1536 HTS [AID873, Type: screening]kallikrein-related peptidase 5 preproprotein [Homo sapiens] [gi:6912644]
View
16
[SID7973802]
 Dose-response cell-based assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID681, Type: confirmatory]Nuclear receptor ROR-alpha [gi:548814]
View
17
[SID7973802]
 Dose-response cell-based assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID681, Type: confirmatory]Nuclear receptor ROR-alpha [gi:548814]
View
18
[SID7973802]
 Dose-response cell-based assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID681, Type: confirmatory]Nuclear receptor ROR-alpha [gi:548814]
View
19
[SID7973802]
 Dose-response cell-based assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID681, Type: confirmatory]Nuclear receptor ROR-alpha [gi:548814]
View
20
[SID7973802]
 Primary Cell-based High Throughput Screening assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID560, Type: screening]Nuclear receptor ROR-alpha [gi:548814]
View
21
[SID7973802]
 Primary Cell-based High Throughput Screening assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID560, Type: screening]Nuclear receptor ROR-alpha [gi:548814]
View
22
[SID7973802]
 Primary Cell-based High Throughput Screening assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID560, Type: screening]Nuclear receptor ROR-alpha [gi:548814]
View
23
[SID7973802]
 Primary Cell-based High Throughput Screening assay for activators of the Retinoic Acid Receptor-related orphan receptor A (RORA) [AID560, Type: screening]Nuclear receptor ROR-alpha [gi:548814]
View
24
[SID7973802]
 Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
View
25
[SID7973802]
 Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
View
26
[SID7973802]
 Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
View
27
[SID7973802]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
View
28
[SID7973802]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
View
29
[SID7973802]
Potency 6.3096qHTS for Agonist of gsp, the Etiologic Mutation Responsible for Fibrous Dysplasia/McCune-Albright Syndrome: qHTS [AID624287, Type: confirmatory]Guanine nucleotide-binding protein G(s) subunit alpha isoforms short [gi:52000961]
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30
[SID7973802]
Potency 10.4179Primary qHTS for delayed death inhibitors of the malarial parasite plastid, 48 hour incubation [AID504832, Type: confirmatory]
View
31
[SID7973802]
Potency 20.7491qHTS Assay for Modulators of miRNAs and/orActivators of miR-21 [AID2288, Type: confirmatory]
View
32
[SID7973802]
IC50 50Kallikrein 5 1536 HTS Dose Response Confirmation [AID1431, Type: confirmatory]kallikrein-related peptidase 5 preproprotein [Homo sapiens] [gi:6912644]
View
33
[SID7973802]
IC50 50Kallikrein 5 1536 HTS Dose Response Confirmation [AID1431, Type: confirmatory]kallikrein-related peptidase 5 preproprotein [Homo sapiens] [gi:6912644]
View
34
[SID7973802]
Potency qHTS Assay for the Inhibitors of L3MBTL1 [AID485360, Type: confirmatory]lethal(3)malignant brain tumor-like protein 1 isoform I [Homo sapiens] [gi:117938328]
View
35
[SID7973802]
Potency qHTS Assay for the Inhibitors of L3MBTL1 [AID485360, Type: confirmatory]lethal(3)malignant brain tumor-like protein 1 isoform I [Homo sapiens] [gi:117938328]
View
36
[SID7973802]
 uHTS Luminescent assay for identification of inhibitors of Sentrin-specific protease 6 (SENP6) [AID2599, Type: screening]SUMO-1-specific protease [Homo sapiens] [gi:6166485]
View
37
[SID7973802]
IC50 uHTS identification of small molecule inhibitors of LYP via a fluorescence intensity assay [AID1779, Type: confirmatory]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
38
[SID7973802]
IC50 uHTS identification of small molecule inhibitors of LYP via a fluorescence intensity assay [AID1779, Type: confirmatory]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
39
[SID7973802]
IC50 uHTS identification of small molecule inhibitors of LYP via a fluorescence intensity assay [AID1779, Type: confirmatory]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
40
[SID7973802]
 HTS for LYP Inhibitors-an Autoimmunity Target - Primary screen [AID606, Type: confirmatory]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
41
[SID7973802]
 HTS for LYP Inhibitors-an Autoimmunity Target - Primary screen [AID606, Type: confirmatory]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
42
[SID7973802]
 HTS for LYP Inhibitors-an Autoimmunity Target - Primary screen [AID606, Type: confirmatory]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
43
[SID7973802]
 LYP Activators-an Autoimmunity Target - Primary screen [AID697, Type: screening]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
44
[SID7973802]
 LYP Activators-an Autoimmunity Target - Primary screen [AID697, Type: screening]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
45
[SID7973802]
 LYP Activators-an Autoimmunity Target - Primary screen [AID697, Type: screening]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
46
[SID7973802]
 LYP Inhibitors-an Autoimmunity Target - Primary screen [AID640, Type: screening]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
47
[SID7973802]
 LYP Inhibitors-an Autoimmunity Target - Primary screen [AID640, Type: screening]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
48
[SID7973802]
 LYP Inhibitors-an Autoimmunity Target - Primary screen [AID640, Type: screening]PTPN22 gene product [Homo sapiens] [gi:224586929]
View
49
[SID7973802]
IC50 uHTS fluorescence polarization assay for the identification of translation initiation inhibitors (PABP) [AID2014, Type: confirmatory]polyadenylate-binding protein 1 [Homo sapiens] [gi:46367787]
View
50
[SID7973802]
 uHTS identification of microRNA-mediated mRNA deadenylation inhibitors by fluoresence polarization assay [AID588489, Type: screening]polyadenylate-binding protein 1 [Homo sapiens] [gi:46367787]
View