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CHEMBL2013231 (CID 59052424) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
BioAssay Types:
Literature(3)
 
 
BioActivity Types:
EC50(2)
 
 
Ki(1)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID160688306]
EC50 0.001Agonist activity at human CXCR7 expressed in HEK293T cells co-expressing beta-arrestin2-YFP assessed as beta-arrestin2 recruitment after 1 hr by BRET assay [AID654455, Type: Literature]Atypical chemokine receptor 3 [gi:115502380]
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2
[SID160688306]
Ki 0.01995Displacement of [125I]-CXCL12 from human CXCR7 expressed in HEK293 cells after 3 hrs [AID654454, Type: Literature]Atypical chemokine receptor 3 [gi:115502380]
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3
[SID160688306]
EC50 0.0237Agonist activity at human CXCR7 expressed in HEK293 cells assessed as reduction of receptor surface expression after 1 hr by ELISA based internalization assay [AID654456, Type: Literature]Atypical chemokine receptor 3 [gi:115502380]
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