CHEMBL1951701 (CID 57402172) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Top Targets:
7TM GPCR Srx(2)
 
 
BioAssay Types:
Literature(3)
 
 
BioActivity Types:
Ki(3)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136942933]
Ki 0.074Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647794, Type: Literature]Mu-type opioid receptor [gi:2851402]
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2
[SID136942933]
Ki 0.074Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647794, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
3
[SID136942933]
Ki 0.074Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647794, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
4
[SID136942933]
Ki 0.074Displacement of [3H]-DAMGO from human mu opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647794, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
5
[SID136942933]
Ki 0.751Displacement of [3H]-U69593 from human kappa opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647796, Type: Literature]Kappa-type opioid receptor [gi:116242691]
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6
[SID136942933]
Ki 0.751Displacement of [3H]-U69593 from human kappa opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647796, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
7
[SID136942933]
Ki 0.751Displacement of [3H]-U69593 from human kappa opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647796, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
8
[SID136942933]
Ki 0.751Displacement of [3H]-U69593 from human kappa opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647796, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
9
[SID136942933]
Ki 5.8Displacement of [3H]-DADLE from human delta opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647795, Type: Literature]Delta-type opioid receptor [gi:311033488]
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10
[SID136942933]
Ki 5.8Displacement of [3H]-DADLE from human delta opioid receptor expressed in CHO cells membrane after 2 hrs by liquid scintillation counting [AID647795, Type: Literature]Delta-type opioid receptor [gi:311033488]
View