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CHEMBL1957717 (CID 57400106) - Compound BioActivity Data
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BioActivity Outcomes:
Active(5)
 
 
Unspecified(1)
 
 
Top Targets:
7tm 4(2)
 
 
BioAssay Types:
Literature(6)
 
 
 
BioActivity Types:
Ki(5)
 
 
Kd(1)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 6    Data Row: 6   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136939235]
Ki 0.0003Antagonist activity at human mu opioid receptor by GTP-gamma S binding assay [AID649256, Type: Literature]Mu-type opioid receptor [gi:2851402]
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2
[SID136939235]
Ki 0.00055Displacement of [3H]DAMGO from mu opioid receptor in dog brain after 90 mins by scintillation counting [AID649261, Type: Literature]
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3
[SID136939235]
Ki 0.00081Displacement of [3H]DAMGO from human mu opioid receptor [AID649258, Type: Literature]Mu-type opioid receptor [gi:2851402]
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4
[SID136939235]
Ki 0.051Displacement of [3H]U-69,593 from kappa opioid receptor in dog brain after 90 mins by scintillation counting [AID649260, Type: Literature]
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5
[SID136939235]
Ki 0.384Displacement of [3H]DPDPE from delta opioid receptor in dog brain after 90 mins by scintillation counting [AID649259, Type: Literature]
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6
[SID136939235]
Kd Antagonist activity at mu opioid receptor in guinea pig longitudinal muscle myenteric plexus assessed as inhibition of DAMGO-induced twitch tension at 1 uM after 10 mins [AID649257, Type: Literature]Mu-type opioid receptor [gi:3024265]
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