CHEMBL1927475 (CID 57397718) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(3)
 
 
Unspecified(1)
 
 
Top Targets:
NR LBD PPAR(3)
 
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
EC50(4)
 
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136934825]
EC50 0.0314Induction of [14C]oleic acid oxidation in a human myotubes after 4 days by beta liquid scintillation counting [AID635193, Type: Literature]
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2
[SID136934825]
EC50 0.58Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635240, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
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3
[SID136934825]
EC50 0.58Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635240, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
View
4
[SID136934825]
EC50 0.58Agonist activity at human PPARdelta ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635240, Type: Literature]Peroxisome proliferator-activated receptor delta [gi:417522]
View
5
[SID136934825]
EC50 0.735Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene assay [AID635238, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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6
[SID136934825]
EC50 0.735Agonist activity at human PPARalpha ligand binding domain expressed in COS-1 cells co-transfected with Gal4 after 24 hrs by luciferase reporter gene assay [AID635238, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
View
7
[SID136934825]
EC50 1Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635239, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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8
[SID136934825]
EC50 1Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635239, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
9
[SID136934825]
EC50 1Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635239, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
10
[SID136934825]
EC50 1Agonist activity at human PPARgamma ligand binding domain expressed in COS-1 cells after 24 hrs by luciferase reporter gene-based luminometeric analysis [AID635239, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View