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CHEMBL1956367 (CID 57395675) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD PPAR(4)
 
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
EC50(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136930882]
EC50 4.9Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648526, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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2
[SID136930882]
EC50 6.6Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648525, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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3
[SID136930882]
Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to Wy-14643 [AID648529, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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4
[SID136930882]
Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to pioglitazone [AID648530, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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