CHEMBL1957843 (CID 57345673) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(5)
 
 
Top Targets:
7TM GPCR Srx(2)
 
 
BioAssay Types:
Literature(5)
 
 
BioActivity Types:
Ki(5)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136932604]
Ki 7e-05Displacement of [3H]DAMGO from mu opioid receptor in dog brain after 90 mins by scintillation counting [AID649261, Type: Literature]
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2
[SID136932604]
Ki 8e-05Antagonist activity at human mu opioid receptor by GTP-gamma S binding assay [AID649256, Type: Literature]Mu-type opioid receptor [gi:2851402]
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3
[SID136932604]
Ki 8e-05Antagonist activity at human mu opioid receptor by GTP-gamma S binding assay [AID649256, Type: Literature]Mu-type opioid receptor [gi:2851402]
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4
[SID136932604]
Ki 8e-05Antagonist activity at human mu opioid receptor by GTP-gamma S binding assay [AID649256, Type: Literature]Mu-type opioid receptor [gi:2851402]
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5
[SID136932604]
Ki 8e-05Antagonist activity at human mu opioid receptor by GTP-gamma S binding assay [AID649256, Type: Literature]Mu-type opioid receptor [gi:2851402]
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6
[SID136932604]
Ki 0.0001Displacement of [3H]DAMGO from human mu opioid receptor [AID649258, Type: Literature]Mu-type opioid receptor [gi:2851402]
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7
[SID136932604]
Ki 0.0001Displacement of [3H]DAMGO from human mu opioid receptor [AID649258, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
8
[SID136932604]
Ki 0.0001Displacement of [3H]DAMGO from human mu opioid receptor [AID649258, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
9
[SID136932604]
Ki 0.0001Displacement of [3H]DAMGO from human mu opioid receptor [AID649258, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
10
[SID136932604]
Ki 0.0045Displacement of [3H]U-69,593 from kappa opioid receptor in dog brain after 90 mins by scintillation counting [AID649260, Type: Literature]
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11
[SID136932604]
Ki 0.019Displacement of [3H]DPDPE from delta opioid receptor in dog brain after 90 mins by scintillation counting [AID649259, Type: Literature]
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