CHEMBL1956364 (CID 57345616) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Unspecified(2)
 
 
Top Targets:
NR LBD PPAR(4)
 
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
EC50(2)
 
 
SAR
Target summary
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136940775]
EC50 0.5Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648526, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
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2
[SID136940775]
EC50 0.5Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648526, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
3
[SID136940775]
EC50 0.5Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648526, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
4
[SID136940775]
EC50 0.5Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648526, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
5
[SID136940775]
EC50 1Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648525, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
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6
[SID136940775]
EC50 1Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay [AID648525, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
View
7
[SID136940775]
 Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to pioglitazone [AID648530, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
8
[SID136940775]
 Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to pioglitazone [AID648530, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
9
[SID136940775]
 Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to pioglitazone [AID648530, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
10
[SID136940775]
 Agonist activity at GAL4-tagged human PPARgamma ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to pioglitazone [AID648530, Type: Literature]Peroxisome proliferator-activated receptor gamma [gi:13432234]
View
11
[SID136940775]
 Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to Wy-14643 [AID648529, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
View
12
[SID136940775]
 Agonist activity at GAL4-tagged human PPARalpha ligand binding domain expressed in HepG2 cells assessed as transactivation after 20 hrs by beta-galactosidase reporter gene assay relative to Wy-14643 [AID648529, Type: Literature]Peroxisome proliferator-activated receptor alpha [gi:3041727]
View