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CHEMBL1934899 (CID 57336563) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Unspecified(2)
 
 
Top Targets:
HDAC8(1)
 
 
HDAC6-dom1(1)
 
 
HDAC1(1)
 
 
HDAC7(1)
 
 
BioAssay Types:
Literature(5)
 
 
 
BioActivity Types:
Kd(5)
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136924745]
Kd 7Inhibition of Bordetella FB188 HDAH using Boc-L-Lys(acetyl)-MCA as substrate by fluorogenic enzymatic assay [AID637887, Type: Literature]
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2
[SID136924745]
Kd 8.2Inhibition of recombinant human HDAC6 using Boc-L-Lys(acetyl)-MCA as substrate by fluorogenic enzymatic assay [AID637889, Type: Literature]Histone deacetylase 6 [gi:205371758]
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3
[SID136924745]
Kd 30Inhibition of recombinant human HDAC7 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assay [AID637890, Type: Literature]Histone deacetylase 7 [gi:30913097]
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4
[SID136924745]
Kd 100Inhibition of recombinant human HDAC1 using Boc-L-Lys(acetyl)-MCA as substrate by fluorogenic enzymatic assay [AID637888, Type: Literature]Histone deacetylase 1 [gi:2498443]
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5
[SID136924745]
Kd 100Inhibition of recombinant human HDAC8 using Boc-L-Lys(trifluoroacetyl)-MCA as substrate by fluorogenic enzymatic assay [AID637891, Type: Literature]Histone deacetylase 8 [gi:29839394]
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