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zolpidem (CID 5732) - Compound BioActivity Data
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BioActivity Outcomes:
Active(179)
 
 
Inactive(231)
 
 
Inconclusive(34)
 
 
Unspecified(184)
 
 
Top Targets:
Neur chan LBD(137)
 
 
 
Neur chan mem..(28)
 
 
 
p450(10)
 
 
 
NR LBD PPAR(8)
 
 
NR LBD ER(7)
 
 
 
BioAssay Types:
Literature(432)
 
 
 
 
 
Confirmatory(149)
 
 
 
 
Summary(24)
 
 
 
 
Screening(18)
 
 
BioActivity Types:
Ki(193)
 
 
 
Potency(161)
 
 
 
 
EC50(12)
 
 
 
IC50(6)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 450    Data Row: 628   Total Pages: 32   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID103238173]
IC50 0.014Inhibition of [3H]flumazenil binding to recombinant GABA-A receptor alpha-1 subunit in cerebellum [AID72469, Type: confirmatory]
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2
[SID103238173]
Ki 0.0155Displacement of [3H]Ro-151788 from benzodiazepine binding site of GABAA alpha-1-beta-2-gamma-2 M130C receptor mutant expressed in HEK293T cells [AID345429, Type: Literature]
View
3
[SID103238173]
Ki 0.019Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cells [AID219782, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:120788]
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4
[SID103238173]
Ki 0.019Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cells [AID219782, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-1 [gi:51317298]
View
5
[SID103238173]
Ki 0.019Binding affinity for rat GABA-A receptor alpha-1-beta-2-gamma-2 subunits expressed in HEK293 cells [AID219782, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-2 [gi:52000957]
View
6
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-2 [gi:52000957]
View
7
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit beta-3 [gi:52000955]
View
8
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit epsilon [gi:13959374]
View
9
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-1 [gi:51317298]
View
10
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-3 [gi:120790]
View
11
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-1 [gi:120782]
View
12
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit gamma-2 [gi:120788]
View
13
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-6 [gi:232127]
View
14
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit delta [gi:544363]
View
15
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit pi [gi:3023821]
View
16
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]GABA theta subunit [gi:81902501]
View
17
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-2 [gi:120758]
View
18
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-3 [gi:120761]
View
19
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-4 [gi:120763]
View
20
[SID103238173]
Ki 0.025Displacement of [3H]- flunitrazepam from rat GABA-A benzodiazepine receptor [AID40372, Type: Literature]Gamma-aminobutyric acid receptor subunit alpha-5 [gi:120764]
View