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CHEMBL1923501 (CID 56926173) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Unspecified(1)
 
 
Top Targets:
Motilin assoc(2)
 
 
BioAssay Types:
Literature(4)
 
 
 
BioActivity Types:
Ki(2)
 
 
EC50(1)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 4    Data Row: 4   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136931425]
Ki 0.086Displacement of [125I-His9]-ghrelin from human GRLN receptor by radioligand binding assay [AID632805, Type: Literature]Appetite-regulating hormone [gi:17865471]
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2
[SID136931425]
EC50 0.134Agonist activity at human GRLN receptor expressed in HEK293 cells assessed as calcium binding by Ca2+ bioluminescence aequorin assay [AID632806, Type: Literature]Appetite-regulating hormone [gi:17865471]
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3
[SID136931425]
Ki Agonist activity at ghrelin receptor [AID711464, Type: Literature]
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4
[SID136931425]
Selectivity ratio of EC50 for mTOR to EC50 for human GRLN receptor [AID632991, Type: Literature]
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