Bookmark and Share
CHEMBL1921841 (CID 56851582) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(3)
 
 
Inactive(3)
 
 
Unspecified(2)
 
 
Top Targets:
7TM GPCR Srx(6)
 
 
 
BioAssay Types:
Literature(8)
 
 
 
 
BioActivity Types:
Ki(3)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 8   Total Pages: 1   
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID136935048]
Ki 0.000622Displacement of [3H]diprenorphine from human opioid kappa receptor expressed in CHO cells after 120 mins by scintillation counting [AID631359, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
2
[SID136935048]
Ki 0.0315Displacement of [3H]diprenorphine from human opioid mu receptor expressed in CHO cells after 120 mins by scintillation counting [AID631360, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
3
[SID136935048]
Ki 0.251Displacement of [3H]diprenorphine from human opioid delta receptor expressed in HEK293 cells after 120 mins by scintillation counting [AID631361, Type: Literature]Delta-type opioid receptor [gi:311033488]
View
4
[SID136935048]
Selectivity ratio of Ki for human opioid mu receptor expressed in CHO cells to Ki for human opioid kappa receptor expressed in CHO cells [AID631362, Type: Literature]
View
5
[SID136935048]
Selectivity ratio of Ki for human opioid delta receptor expressed in HEK293 cells to Ki for human opioid kappa receptor expressed in CHO cells [AID631363, Type: Literature]
View
6
[SID136935048]
Agonist activity at human opioid mu receptor expressed in CHO cells assessed as stimulation of [35S]-GTPgammaS binding at 10 uM [AID631393, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
7
[SID136935048]
Agonist activity at human opioid delta receptor expressed in HEK293 cells assessed as stimulation of [35S]-GTPgammaS binding at 10 uM [AID631394, Type: Literature]Delta-type opioid receptor [gi:311033488]
View
8
[SID136935048]
Agonist activity at human opioid kappa receptor expressed in CHO cells assessed as stimulation of [35S]-GTPgammaS binding at 10 uM [AID631392, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View