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BRD-K95932625-001-01-8 (CID 56840711) - Compound BioActivity Data
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BioActivity Outcomes:
Active(3)
 
 
Inactive(9)
 
 
Inconclusive(2)
 
 
Unspecified(1)
 
 
Top Targets:
PKc like(4)
 
 
 
STKc CDK5(1)
 
 
CDK5 activato..(1)
 
 
BioAssay Types:
Confirmatory(7)
 
 
 
 
BioActivity Types:
AC50(7)
 
 
 
 
IC50(6)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 8    Data Row: 15   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134970448]
AC50_uM 5.57GSK3beta Measured in Biochemical System Using Plate Reader - 2046-01_Inhibitor_Dose_DryPowder_Activity [AID623998, Type: confirmatory]glycogen synthase kinase-3 beta isoform 1 [Homo sapiens] [gi:21361340]
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2
[SID134970448]
AC50_uM 31.91GSK3beta Assay at Varied ATP concentrations Measured in Biochemical System Using Plate Reader - 2046-04_Inhibitor_Dose_DryPowder_Activity [AID624027, Type: confirmatory]glycogen synthase kinase-3 beta isoform 1 [Homo sapiens] [gi:21361340]
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3
[SID134970448]
GSK3beta Surface Plasmon Resonance (SPR) Assay Measured in Biochemical System Using Microfluidics - 2133-08_Inhibitor_Dose_DryPowder_Activity [AID624108, Type: other]glycogen synthase kinase-3 beta isoform 1 [Homo sapiens] [gi:21361340]
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4
[SID134970448]
Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091, Type: other]glycogen synthase kinase-3 beta isoform 1 [Homo sapiens] [gi:21361340]
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5
[SID134970448]
GSK3a IC50 1.24173Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091_5, Type: other]
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6
[SID134970448]
GSK3b IC50 2.71971Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091_6, Type: other]
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7
[SID134970448]
CDC2/CycB1 IC50 10Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091_1, Type: other]
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8
[SID134970448]
CDK2/CycA2 IC50 10Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091_2, Type: other]
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9
[SID134970448]
CDK2/CycE1 IC50 10Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091_3, Type: other]
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10
[SID134970448]
CDK5/p25 IC50 10Dose responses of selected compounds against GSK3b Measured in Biochemical System Using Plate Reader - 2133-10_Inhibitor_Dose_DryPowder_Activity [AID624091_4, Type: other]
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11
[SID134970448]
AC50_uM 35Human p-Tau and Total Tau ELISA Measured in Cell-Based System Using Plate Reader - 2133-07_Inhibitor_Dose_DryPowder_Activity [AID624057, Type: confirmatory]
View
12
[SID134970448]
AC50_uM TCF/LEF Reporter Assay Measured in Cell-Based System Using Plate Reader - 2133-01_Inhibitor_Dose_DryPowder_Activity [AID624086, Type: confirmatory]
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13
[SID134970448]
AC50_uM PathHunter bCatenin (U2-OS) Measured in Cell-Based System Using Plate Reader - 2133-06_Inhibitor_Dose_DryPowder_Activity [AID624088, Type: confirmatory]
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14
[SID134970448]
AC50_uM CDK5 Measured in Biochemical System Using Plate Reader - 2046-05_Inhibitor_Dose_DryPowder_Activity [AID623999, Type: confirmatory]Cyclin-dependent kinase 5, regulatory subunit 1 (p35) [Homo sapiens] [gi:20072248]
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15
[SID134970448]
AC50_uM CDK5 Measured in Biochemical System Using Plate Reader - 2046-05_Inhibitor_Dose_DryPowder_Activity [AID623999, Type: confirmatory]CDK5 [Homo sapiens] [gi:48146199]
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