CHEMBL1790575
(CID
56682530
) -
BioAssay Data Summary for Compound
.
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BioActivity Outcomes:
Active(4)
BioAssay Types:
Literature(
4
)
BioActivity Types:
Ki(
4
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 4 Data Row: 4 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
134462314
]
Active
Ki
0.00042
Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors [AID
217360
, Type: Literature]
View
X
Row No.
1
Structure
Substance
SID
134462314
CID
56682530
Outcome
Active
Ki
0.00042 [uM]
BioAssay
Binding affinity against human vasopressin V1b receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors
AID
217360
BioAssay type
Literature
Target
PubMed
15084136
Data Table
2
[SID
134462314
]
Active
Ki
0.0099
Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors [AID
217394
, Type: Literature]
View
X
Row No.
2
Structure
Substance
SID
134462314
CID
56682530
Outcome
Active
Ki
0.0099 [uM]
BioAssay
Binding affinity against human vasopressin V2 receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors
AID
217394
BioAssay type
Literature
Target
PubMed
15084136
Data Table
3
[SID
134462314
]
Active
Ki
0.0168
Binding affinity against human vasopressin V1a receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors [AID
217087
, Type: Literature]
View
X
Row No.
3
Structure
Substance
SID
134462314
CID
56682530
Outcome
Active
Ki
0.0168 [uM]
BioAssay
Binding affinity against human vasopressin V1a receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors
AID
217087
BioAssay type
Literature
Target
PubMed
15084136
Data Table
4
[SID
134462314
]
Active
Ki
0.102
Binding affinity against human oxytocin receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors [AID
151798
, Type: Literature]
View
X
Row No.
4
Structure
Substance
SID
134462314
CID
56682530
Outcome
Active
Ki
0.102 [uM]
BioAssay
Binding affinity against human oxytocin receptor was determined by using plasma membranes from CHO cells stably transfected with VP/OT receptors
AID
151798
BioAssay type
Literature
Target
PubMed
15084136
Data Table