CHEMBL1834416 (CID 56681955) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(4)
 
 
Unspecified(5)
 
 
Top Targets:
7TM GPCR Srx(4)
 
 
 
BioAssay Types:
Literature(9)
 
 
 
BioActivity Types:
Ki(4)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 9    Data Row: 9   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134461398]
Ki 0.00867Displacement of [3H]Cl-DPDPE from human DOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621888, Type: Literature]Delta-type opioid receptor [gi:311033488]
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2
[SID134461398]
Ki 0.00867Displacement of [3H]Cl-DPDPE from human DOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621888, Type: Literature]Delta-type opioid receptor [gi:311033488]
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3
[SID134461398]
Ki 0.0105Displacement of [3H]DAMGO from human MOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621887, Type: Literature]Mu-type opioid receptor [gi:2851402]
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4
[SID134461398]
Ki 0.0105Displacement of [3H]DAMGO from human MOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621887, Type: Literature]Mu-type opioid receptor [gi:2851402]
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5
[SID134461398]
Ki 0.0105Displacement of [3H]DAMGO from human MOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621887, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
6
[SID134461398]
Ki 0.0105Displacement of [3H]DAMGO from human MOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621887, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
7
[SID134461398]
Ki 0.0355Displacement of [3H]U69593 from human KOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621889, Type: Literature]Kappa-type opioid receptor [gi:116242691]
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8
[SID134461398]
Ki 0.0355Displacement of [3H]U69593 from human KOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621889, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
9
[SID134461398]
Ki 0.0355Displacement of [3H]U69593 from human KOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621889, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
10
[SID134461398]
Ki 0.0355Displacement of [3H]U69593 from human KOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621889, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
11
[SID134461398]
Ki 0.159Displacement of [3H]N/OFQ from human NOP receptor expressed in CHO cells after 60 mins by scintillation counting [AID621019, Type: Literature]Nociceptin receptor [gi:730230]
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12
[SID134461398]
 Partial agonist activity at human NOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to nociceptin [AID621028, Type: Literature]Nociceptin receptor [gi:730230]
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13
[SID134461398]
 Selectivity ratio of Ki for human MOP receptor to Ki for human NOP receptor [AID621020, Type: Literature]
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14
[SID134461398]
 Partial agonist activity at human DOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to DPDPE [AID621026, Type: Literature]Delta-type opioid receptor [gi:311033488]
View
15
[SID134461398]
 Partial agonist activity at human DOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to DPDPE [AID621026, Type: Literature]Delta-type opioid receptor [gi:311033488]
View
16
[SID134461398]
 Partial agonist activity at human KOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to U69593 [AID621027, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
17
[SID134461398]
 Partial agonist activity at human KOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to U69593 [AID621027, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
18
[SID134461398]
 Partial agonist activity at human KOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to U69593 [AID621027, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
19
[SID134461398]
 Partial agonist activity at human KOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to U69593 [AID621027, Type: Literature]Kappa-type opioid receptor [gi:116242691]
View
20
[SID134461398]
 Partial agonist activity at human MOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to DAMGO [AID621025, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
21
[SID134461398]
 Partial agonist activity at human MOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to DAMGO [AID621025, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
22
[SID134461398]
 Partial agonist activity at human MOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to DAMGO [AID621025, Type: Literature]Mu-type opioid receptor [gi:2851402]
View
23
[SID134461398]
 Partial agonist activity at human MOP receptor expressed in CHO cells assessed as maximal stimulation of [35S]GTPgammaS binding after 60 mins by scintillation counting relative to DAMGO [AID621025, Type: Literature]Mu-type opioid receptor [gi:2851402]
View