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CHEMBL1818335 (CID 56676328) - Compound BioActivity Data
.
BioActivity Outcomes:
Active(2)
 
 
Unspecified(3)
 
 
Top Targets:
7tm 4(2)
 
 
BioAssay Types:
Literature(5)
 
 
 
BioActivity Types:
Ki(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 5    Data Row: 5   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134455172]
Ki 0.009Agonist activity at human kappa opioid receptor by GTPgamma S binding assay [AID613670, Type: Literature]Kappa-type opioid receptor [gi:116242691]
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2
[SID134455172]
Ki 0.021Agonist activity at human mu opioid receptor by GTPgamma S binding assay [AID613671, Type: Literature]Mu-type opioid receptor [gi:2851402]
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3
[SID134455172]
Intrinsic clearance in human liver microsomes [AID613643, Type: Literature]
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4
[SID134455172]
Efflux ratio of permeability from basolateral to apical side over apical to basolateral side in MDCK cells expressing human MDR1 [AID613644, Type: Literature]
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5
[SID134455172]
Selectivity, ratio of Ki for human mu opioid receptor to Ki for human kappa opioid receptor [AID613646, Type: Literature]
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