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CHEMBL2431129 (CID 56593278) - Compound BioActivity Data
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BioActivity Outcomes:
Active(2)
 
 
Inactive(1)
 
 
Unspecified(3)
 
 
Top Targets:
7tm 4(3)
 
 
 
BioAssay Types:
Literature(4)
 
 
 
Confirmatory(2)
 
 
 
BioActivity Types:
EC50(5)
 
 
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 6    Data Row: 6   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134225048]
EC50_Mean 4.1SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID602356, Type: confirmatory]neurotensin receptor type 1 [Homo sapiens] [gi:110611243]
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2
[SID174498739]
EC50 4.1Agonist activity at NTR1 (unknown origin) expressed in human U2OS cells coexpressing beta-arrestin by GFP reporter gene assay [AID772307, Type: Literature]Neurotensin receptor type 1 [gi:62297312]
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3
[SID174498739]
EC50 40Agonist activity at GPR35 (unknown origin) expressed in human U2OS cells coexpressing beta-arrestin by GFP reporter gene assay [AID772304, Type: Literature]G-protein coupled receptor 35 [gi:68068087]
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4
[SID174498739]
EC50 80Agonist activity at NTR2 (unknown origin) expressed in human U2OS cells coexpressing beta-arrestin by GFP reporter gene assay [AID772305, Type: Literature]Neurotensin receptor type 2 [gi:311033404]
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5
[SID174498739]
Agonist activity at NTR1 (unknown origin) expressed in human U2OS cells coexpressing beta-arrestin by GFP reporter gene assay relative to neurotensin (8 to 13) [AID772306, Type: Literature]Neurotensin receptor type 1 [gi:62297312]
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6
[SID134225048]
EC50_Mean 80SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID602334, Type: confirmatory]neurotensin receptor type 2 [Homo sapiens] [gi:6912538]
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