MLS-0471472.0001
(CID
56593274
) -
BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Inactive(
2
)
BioAssay Types:
Confirmatory(
2
)
BioActivity Types:
EC50(
2
)
SAR
Target summary
Data download
Chemical Probe
Active
Inactive
Inconclusive
Unspecified
Total Bioassays: 2 Data Row: 2 Total Pages: 1
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#
Substance
Activity
BioAssay
Target
Links
Outcome
Type
Value [μM]
1
[SID
134225038
]
Inactive
EC50
80
SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID
602356
, Type: confirmatory]
NTSR1 gene product [Homo sapiens] [gi:
110611243
]
View
X
Row No.
1
Structure
Substance
SID
134225038
CID
56593274
Outcome
Inactive
EC50
80 [uM]
BioAssay
SAR analysis of small molecule Agonists NTR1 in a image based assay set 3
AID
602356
BioAssay type
confirmatory
Target
NTSR1 gene product [Homo sapiens] [gi:
110611243
]
PubMed
Data Table
2
[SID
134225038
]
Inactive
EC50
80
SAR analysis of small molecule Agonists NTR1 in a image based assay set 3 [AID
602356
, Type: confirmatory]
NTSR1 gene product [Homo sapiens] [gi:
110611243
]
View
X
Row No.
2
Structure
Substance
SID
134225038
CID
56593274
Outcome
Inactive
EC50
80 [uM]
BioAssay
SAR analysis of small molecule Agonists NTR1 in a image based assay set 3
AID
602356
BioAssay type
confirmatory
Target
NTSR1 gene product [Homo sapiens] [gi:
110611243
]
PubMed
Data Table
3
[SID
134225038
]
Inactive
EC50
80
SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID
602334
, Type: confirmatory]
NTSR2 gene product [Homo sapiens] [gi:
6912538
]
View
X
Row No.
3
Structure
Substance
SID
134225038
CID
56593274
Outcome
Inactive
EC50
80 [uM]
BioAssay
SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2
AID
602334
BioAssay type
confirmatory
Target
NTSR2 gene product [Homo sapiens] [gi:
6912538
]
PubMed
Data Table
4
[SID
134225038
]
Inactive
EC50
80
SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2 [AID
602334
, Type: confirmatory]
NTSR2 gene product [Homo sapiens] [gi:
6912538
]
View
X
Row No.
4
Structure
Substance
SID
134225038
CID
56593274
Outcome
Inactive
EC50
80 [uM]
BioAssay
SAR analysis of small molecule NTR1 agonists in a image based NTR2 selectivity assay set 2
AID
602334
BioAssay type
confirmatory
Target
NTSR2 gene product [Homo sapiens] [gi:
6912538
]
PubMed
Data Table