Morpholino(4-phenyl-2H-1,2,3-triazol-2-yl)methanone (CID 56593038) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(5)
 
 
Inactive(8)
 
 
Top Targets:
Peptidase S9(4)
 
 
 
PRK11460(3)
 
 
PGAP1(2)
 
 
PLN02442(2)
 
 
 
Lipase 3(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 13   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_3, Type: other]Abhydrolase domain containing 11 [Mus musculus] [gi:47682716]
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2
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_3, Type: other]Abhydrolase domain containing 11 [Mus musculus] [gi:47682716]
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3
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_4, Type: other]Esterase D/formylglutathione hydrolase [Mus musculus] [gi:55777188]
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4
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_4, Type: other]Esterase D/formylglutathione hydrolase [Mus musculus] [gi:55777188]
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5
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_5, Type: other]Apeh protein [Mus musculus] [gi:20072022]
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6
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_5, Type: other]Apeh protein [Mus musculus] [gi:20072022]
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7
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAFAH2: Fluorescence-based biochemical gel-based Activity-Based Protein Profiling (ABPP) inhibition and selectivity [AID504513_3, Type: other]Abhydrolase domain containing 11 [Mus musculus] [gi:47682716]
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8
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAFAH2: Fluorescence-based biochemical gel-based Activity-Based Protein Profiling (ABPP) inhibition and selectivity [AID504513_1, Type: other]platelet-activating factor acetylhydrolase 2, cytoplasmic [Mus musculus] [gi:225579137]
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9
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAFAH2: Fluorescence-based biochemical gel-based Activity-Based Protein Profiling (ABPP) inhibition and selectivity [AID504513_4, Type: other]Esterase D/formylglutathione hydrolase [Mus musculus] [gi:55777188]
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10
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAFAH2: Fluorescence-based biochemical gel-based Activity-Based Protein Profiling (ABPP) inhibition and selectivity [AID504513_5, Type: other]Lypla1 [Mus musculus] [gi:71059731]
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11
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of overexpressed DAGLb in vitro; triazole urea library [AID602303, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
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12
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of diacylglycerol lipase, beta (DAGLb): fluorescence-based biochemical gel-based competitive Activity-Based Protein Profiling (ABPP) inhibition of overexpressed DAGLb in vitro; triazole urea library [AID602303, Type: other]Daglb gene product [Mus musculus] [gi:31559956]
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13
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAFAH2: Fluorescence-based biochemical gel-based Activity-Based Protein Profiling (ABPP) inhibition and selectivity [AID504513, Type: other]platelet-activating factor acetylhydrolase 2, cytoplasmic [Mus musculus] [gi:225579137]
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14
[SID99445324]
 Late stage assay provider results from the probe development effort to identify inhibitors of PAFAH2: Fluorescence-based biochemical gel-based Activity-Based Protein Profiling (ABPP) inhibition and selectivity [AID504513_2, Type: other]Apeh protein [Mus musculus] [gi:20072022]
View
15
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_1, Type: other]Lypla1 [Mus musculus] [gi:71059731]
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16
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_1, Type: other]Lypla1 [Mus musculus] [gi:71059731]
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17
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111, Type: other]Lypla1 [Mus musculus] [gi:71059731]
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18
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111, Type: other]Lypla1 [Mus musculus] [gi:71059731]
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19
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_2, Type: other]lysophospholipase 2 [Mus musculus] [gi:123122209]
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20
[SID99445324]
 Late stage assay provider results from the probe development effort to identify dual inhibitors of LYPLA1 and LYPLA2: Fluorescence-based biochemical gel-based ABPP inhibition and selectivity [AID493111_2, Type: other]lysophospholipase 2 [Mus musculus] [gi:123122209]
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