STK619281 (CID 5504281) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Inactive(23)
 
 
Top Targets:
crotonase-lik..(1)
 
 
UBCc(1)
 
 
SET(1)
 
 
Rapamycin bin..(1)
 
 
RNA dep RNAP(1)
 
 
BioAssay Types:
Screening(8)
 
 
Literature(2)
 
 
Confirmatory(1)
 
 
SAR
Target summary
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 23    Data Row: 23   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID11535089]
 NMR Based Screening Assay for Influenza A RNA Promoter [AID1637, Type: other]
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2
[SID49808135]
 High Throughput Screen of 100,000 compound library to Identify Inhibitors of Mycobacterium tuberculosis H37Rv [AID1949, Type: confirmatory]
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3
[SID85826973]
 Luminescence Cell-Based Primary HTS to Measure Viability of BJeLR cells [AID2275, Type: screening]
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4
[SID85826973]
 Fluorescence Cell-Based Primary HTS to Identify Reactive Oxygen Species Inducers in Cancer Cells Measured in Cell-Based System Using Plate Reader and Imaging Combination - 2044-01_Activator_SinglePoint_HTS_Activity [AID624156, Type: screening]
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5
[SID85826973]
 Luminescence Cell-Based Primary HTS to Identify Re-Activators of the P53 Mutant Pathway Measured in Cell-Based System Using Plate Reader - 2071-01_Activator_SinglePoint_HTS_Activity [AID624151, Type: screening]
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6
[SID11535089]
 NMR Based Screening Assay for the substrate binding domain of the chaperone DnaK [AID1033, Type: screening]DnaK protein homolog [Escherichia coli] [gi:216546]
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7
[SID92182424]
 A screen for compounds that inhibit processive DNA synthesis of vaccinia virus [AID493162, Type: other]DNA polymerase [Vaccinia virus] [gi:335756]
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8
[SID92182424]
 A screen for compounds that inhibit the bacterial siderophore biosynthetic enzyme MbtI [AID493033, Type: other]Isochorismate synthase/isochorismate-pyruvate lyase mbtI [gi:81706979]
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9
[SID11535089]
 NMR Based Screening Assay for Novel Chemotypes against influenza A virus [AID1549, Type: other]M2 [Influenza A virus (A/TW/4845/1999(H1N1))] [gi:89033149]
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10
[SID92182424]
 A screen for compounds that inhibit viral RNA polymerase binding and polymerization activities [AID588519, Type: Literature]Chain A, Poliovirus Polymerase With Gtp [gi:52695378]
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11
[SID11535089]
 NMR Based Screening Assay For Novel Chemical Probes Targeting The FRB Domain of mTOR [AID1648, Type: other]Chain A, Nmr Solution Structure Of The Frb Domain Of Mtor [gi:159164579]
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12
[SID85826973]
 EZH2/PRC2 methyltransferase inhibitors Measured in Biochemical System Using Plate Reader - 2125-01_Inhibitor_SinglePoint_HTS_Activity [AID651548, Type: screening]EZH2 gene product [Homo sapiens] [gi:21361095]
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13
[SID11535089]
 NMR Based Screening Assay for FKBP12 [AID608, Type: other]peptidyl-prolyl cis-trans isomerase FKBP1A isoform a [Homo sapiens] [gi:17149836]
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14
[SID11535089]
 NMR Based Screening Assay for FKBP12 [AID608, Type: other]peptidyl-prolyl cis-trans isomerase FKBP1A isoform a [Homo sapiens] [gi:17149836]
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15
[SID85826973]
 SMM ID4 Measured in Biochemical System Using Small Molecule MicroArray - 2128-01_Other_SinglePoint_HTS_Activity [AID624137, Type: screening]Id4 [Homo sapiens] [gi:881546]
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16
[SID85826973]
 Development of IDH1/2 inhibitors (CTD2project) Measured in Biochemical System Using Plate Reader - 2107-01_Inhibitor_SinglePoint_HTS_Activity [AID624101, Type: screening]Isocitrate dehydrogenase 1 (NADP+), soluble [Homo sapiens] [gi:62203298]
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17
[SID85826973]
 Development of IDH1/2 inhibitors (CTD2project) Measured in Biochemical System Using Plate Reader - 2107-01_Inhibitor_SinglePoint_HTS_Activity [AID624101, Type: screening]Isocitrate dehydrogenase 1 (NADP+), soluble [Homo sapiens] [gi:62203298]
View
18
[SID85826973]
 Development of IDH1/2 inhibitors (CTD2project) Measured in Biochemical System Using Plate Reader - 2107-01_Inhibitor_SinglePoint_HTS_Activity [AID624101, Type: screening]Isocitrate dehydrogenase 1 (NADP+), soluble [Homo sapiens] [gi:62203298]
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19
[SID11535089]
 NMR assay targeting the ubiquitin-proteasome system to modulate protein folding and degradation [AID1552, Type: other]UBE2N gene product [Homo sapiens] [gi:4507793]
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20
[SID11535089]
 NMR assay targeting the ubiquitin-proteasome system to modulate protein folding and degradation [AID1552, Type: other]UBE2N gene product [Homo sapiens] [gi:4507793]
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21
[SID85826973]
 NSD2 Inhibitors Measured in Biochemical System Using Plate Reader - 2115-01_Inhibitor_SinglePoint_HTS_Activity [AID624260, Type: screening]WHSC1 gene product [Homo sapiens] [gi:109633019]
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22
[SID124869491]
 A screen for small molecule inhibitors of the human deubiquitinating enzyme, UCH37 [AID588478, Type: other]ubiquitin C-terminal hydrolase UCH37 [Homo sapiens] [gi:4877999]
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23
[SID92182424]
 A screen for compounds that inhibit the MenB enzyme of Mycobacterium tuberculosis [AID540299, Type: Literature]naphthoate synthase [Mycobacterium tuberculosis H37Rv] [gi:15607688]
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24
[SID92182424]
 A screen for compounds that inhibit replication of Vibrio cholerae chromosome II [AID504770, Type: other]hypothetical protein VC_A0002 [Vibrio cholerae O1 biovar El Tor str. N16961] [gi:9657380]
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25
[SID92182424]
 A screen for compounds that inhibit the CapD enzyme of Bacillus anthracis [AID492967, Type: other]gamma-glutamyltranspeptidase [Bacillus anthracis str. 'Ames Ancestor'] [gi:47566732]
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26
[SID92182424]
 A screen for compounds that inhibit the activity of Staphylococcus aureus DNA helicase [AID485395, Type: other]replicative DNA helicase [Staphylococcus aureus subsp. aureus JH1] [gi:150392496]
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27
[SID92182424]
 A screen for compounds that modulate the activity of the Staphylococcus aureus MgrA protein [AID602314, Type: other]MarR family regulatory protein [Staphylococcus aureus subsp. aureus str. Newman] [gi:151220867]
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