CHEMBL1819172 (CID 54768920) - BioAssay Data Summary for Compound
.
BioActivity Outcomes:
Active(2)
 
 
Unspecified(1)
 
 
Top Targets:
Esterase lipa..(2)
 
 
BioAssay Types:
Literature(3)
 
 
 
BioActivity Types:
IC50(2)
 
 
SAR
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID134442496]
IC50 0.034Inhibition of human serum recombinant AChE using acetylthiocholine iodide as substrate preincubated for 20 mins by Ellman's method [AID613944, Type: Literature]Acetylcholinesterase [gi:113037]
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2
[SID134442496]
IC50 0.0381Inhibition of human serum recombinant BChE using butyrylthiocholine iodide as substrate preincubated for 20 mins by Ellman's method [AID613945, Type: Literature]Cholinesterase [gi:116353]
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3
[SID134442496]
 Selectivity ratio of IC50 for human serum recombinant BuChE to IC50 for human serum recombinant AChE [AID613946, Type: Literature]
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