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NSC675805 (CID 54680429) - Compound BioActivity Data
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BioActivity Outcomes:
Active(8)
 
 
Inactive(804)
 
 
Inconclusive(6)
 
 
Unspecified(5)
 
 
Top Targets:
7tm 4(43)
 
 
alkPPc(12)
 
 
Bcl-2 like(11)
 
 
Tryp SPc(9)
 
 
G-alpha(8)
 
 
 
BioAssay Types:
Screening(514)
 
 
 
 
 
Confirmatory(273)
 
 
 
 
 
Literature(13)
 
 
BioActivity Types:
Potency(150)
 
 
 
 
 
IC50(53)
 
 
 
EC50(10)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 748    Data Row: 823   Total Pages: 42   Display: Page     
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID14723641]
Potency 14.1254qHTS Assay for Activators of ClpP [AID651965, Type: confirmatory]ClpP [Bacillus subtilis] [gi:2668494]
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2
[SID14723641]
uHTS identification of inhibitors of cullin neddylation in a TR-FRET assay [AID651699, Type: screening]NEDD8-activating enzyme E1 regulatory subunit isoform a [Homo sapiens] [gi:4502169]
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3
[SID14723641]
uHTS identification of inhibitors of cullin neddylation in a TR-FRET assay [AID651699, Type: screening]NEDD8-conjugating enzyme Ubc12 [Homo sapiens] [gi:4507791]
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4
[SID14723641]
uHTS identification of modulators of interaction between CendR and NRP-1 using Fluorescence Polarization assay [AID602438, Type: screening]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
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5
[SID14723641]
Fluorescence-based biochemical primary high throughput screening assay to identify inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis [AID588726, Type: screening]fructose-bisphosphate aldolase [Mycobacterium tuberculosis H37Rv] [gi:15607504]
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6
[SID14723641]
Fluorescence-based biochemical high throughput confirmation assay for inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis [AID651616, Type: screening]fructose-bisphosphate aldolase [Mycobacterium tuberculosis H37Rv] [gi:15607504]
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7
[SID14723641]
Primary HTS assay for chemical inhibitors of TNF alpha stimulated E-Selectin expression [AID1246, Type: screening]selectin E [Homo sapiens] [gi:56417702]
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8
[SID14723641]
Counterscreen for inhibitors of the fructose-bisphosphate aldolase (FBA) of M. tuberculosis: Fluroescence-based biochemical high throughput Glycerophosphate Dehydrogenase-Triosephosphate Isomerase (GDH-TPI) assay to identify assay artifacts [AID652141, Type: screening]
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9
[SID14723641]
IC50_1_FP 95Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay [AID651650_2, Type: confirmatory]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
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10
[SID14723641]
IC50_2_FP 95Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay [AID651650_3, Type: confirmatory]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
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11
[SID14723641]
IC50_1_AlphaScreen 100Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay [AID651650_5, Type: confirmatory]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
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12
[SID14723641]
Potency qHTS for Inhibitors of Human Acid Sphingomyelinase Assay: Native Substrate [AID624178, Type: confirmatory]acid sphingomyelinase [Homo sapiens] [gi:179095]
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13
[SID14723641]
Assay for HTS of Gi/Go-linked GPCRs using mGluR8: Primary Screening [AID488969, Type: screening]metabotropic glutamate receptor 8 [Rattus norvegicus] [gi:1575471]
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14
[SID14723641]
IC50_CUL1 neddylation_Mean 48Dose-response confirmation of inhibitors of cullin neddylation in a TR-FRET assay [AID652247, Type: confirmatory]NEDD8-activating enzyme E1 regulatory subunit isoform a [Homo sapiens] [gi:4502169]
View
15
[SID14723641]
IC50_CUL1 neddylation_Mean 48Dose-response confirmation of inhibitors of cullin neddylation in a TR-FRET assay [AID652247, Type: confirmatory]NEDD8-conjugating enzyme Ubc12 [Homo sapiens] [gi:4507791]
View
16
[SID14723641]
Potency 56.2341qHTS Assay for Substrates of Mammalian Selenoprotein Thioredoxin Reductase 1 (TrxR1): qHTS [AID588456, Type: confirmatory]thioredoxin reductase [Rattus norvegicus] [gi:8659577]
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17
[SID14723641]
Potency 89.1251HTS for Inhibitors of HP1-beta Chromodomain Interactions with Methylated Histone Tails [AID540317, Type: confirmatory]chromobox protein homolog 1 [Homo sapiens] [gi:187960037]
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18
[SID14723641]
IC50_FP_Mean 95Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay [AID651650, Type: confirmatory]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
View
19
[SID14723641]
IC50_FP_Mean 95Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay [AID651650_1, Type: confirmatory]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
View
20
[SID14723641]
IC50_AlphaScreen_Mean 100Dose Response confirmation of small molecule modulators of the interaction between CendR and NRP-1 in a panel assay [AID651650_4, Type: confirmatory]Chain A, Crystal Structure Of The B1b2 Domains From Human Neuropilin-1 [gi:160877737]
View