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BioActivity Data for Compound Scandenin (CID 54676535)

BioActivity Outcomes:
Active(5)
 
 
Inactive(79)
 
 
Inconclusive(9)
 
 
Unspecified(36)
 
 
Top Targets:
PLDc mTdp1 2(3)
 
 
P53(2)
 
 
NR LBD TR(2)
 
 
NR LBD ROR li..(2)
 
 
Menin(2)
 
 
BioAssay Types:
Confirmatory(69)
 
 
 
 
Literature(42)
 
 
 
 
Screening(13)
 
 
 
BioAssay Categories:
In vitro(6)
 
 
 
Toxicity(4)
 
 
 
ADME(6)
 
 
 
Cell-based(14)
 
 
 
 
 
BioActivity Types:
Potency(67)
 
 
 
 
IC50(2)
 
 
Ki(2)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 124    Data Row: 129   Total Pages: 7   Display: Page     
Sort: [Click the result table header to sort]
#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID174510284]
Ki 0.56Ki values for sodium fluorescein (10 uM) uptake in OATP1B3-transfected CHO cells [AID977604, Type: Literature]
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2
[SID174510284]
Ki 0.59Ki values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cells [AID977601, Type: Literature]
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3
[SID174510284]
IC50 0.74131pIC50 values for sodium fluorescein (10 uM) uptake in OATP1B3-transfected CHO cells [AID977603, Type: Literature]
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4
[SID174510284]
IC50 1.07152pIC50 values for sodium fluorescein (10 uM) uptake in OATP1B1-transfected CHO cells [AID977600, Type: Literature]
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5
[SID26749607]
Potency 79.4328Inhibitors of USP1/UAF1: Pilot qHTS [AID504865, Type: confirmatory]USP1 protein, partial [Homo sapiens] [gi:118600387]
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6
[SID174510284]
Insecticidal activity against Achaea janata assessed as larval duration at 4 ug/larva administered through topical application (Rvb = 7.3 +/- 0.1 days) [AID1104290, Type: Literature]
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7
[SID174510284]
Insecticidal activity against Achaea janata assessed as larval duration at 2 ug/larva administered through topical application (Rvb = 7.3 +/- 0.1 days) [AID1104291, Type: Literature]
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8
[SID174510284]
Inhibition of sodium fluorescein uptake in OATP1B3-transfected CHO cells at an equimolar substrate-inhibitor concentration of 10 uM [AID977602, Type: Literature]
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9
[SID174510284]
Insecticidal activity against 3 to 8 days old Callosobruchus chinensis assessed as mortality at 1 ug/mL measured after 24 hr by fumigation assay [AID1081936, Type: Literature]
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10
[SID174510284]
Insecticidal activity against Achaea janata assessed as adult emergence at 2 ug/larva administered through topical application (Rvb = 98.8 +/- 0.5 %) [AID1104277, Type: Literature]
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11
[SID174510284]
Inhibition of sodium fluorescein uptake in OATP1B1-transfected CHO cells at an equimolar substrate-inhibitor concentration of 10 uM [AID977599, Type: Literature]
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12
[SID174510284]
Insecticidal activity against Achaea janata assessed as adult deformity at 2 ug/larva administered through topical application [AID1104279, Type: Literature]
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13
[SID174510284]
Insecticidal activity against Achaea janata assessed as adult deformity at 4 ug/larva administered through topical application [AID1104280, Type: Literature]
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14
[SID174510284]
Insecticidal activity against Achaea janata assessed as pupal mortality at 4 ug/larva administered through topical application [AID1104282, Type: Literature]
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15
[SID174510284]
Insecticidal activity against Achaea janata assessed as pupal weight at 2 ug/larva administered through topical application (Rvb = 696.4 +/- 2.6 mg) [AID1104283, Type: Literature]
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16
[SID174510284]
Insecticidal activity against Achaea janata assessed as pupal weight at 4 ug/larva administered through topical application (Rvb = 696.4 +/- 2.6 mg) [AID1104284, Type: Literature]
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17
[SID174510284]
Insecticidal activity against Achaea janata assessed as pupal duration at 2 ug/larva administered through topical application (Rvb = 10.3 +/- 0.1 days) [AID1104285, Type: Literature]
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18
[SID174510284]
Insecticidal activity against Achaea janata assessed as larval mortality at 4 ug/larva administered through topical application [AID1104288, Type: Literature]
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19
[SID174510284]
Insecticidal activity against Achaea janata assessed as larval mortality at 2 ug/larva administered through topical application [AID1104289, Type: Literature]
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20
[SID174510284]
Toxicity against Achaea janata at 10 ug/cm2 after 24 hr by leaf disk method [AID1104292, Type: Literature]
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