CHEMBL1783515 (CID 54584310) - BioAssay Data Summary for Compound
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BioActivity Outcomes:
Active(3)
 
 
Top Targets:
Esterase lipa..(3)
 
 
BioAssay Types:
Literature(3)
 
 
BioActivity Types:
IC50(3)
 
 
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Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 3    Data Row: 3   Total Pages: 1   
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OutcomeTypeValue [μM]
1
[SID131280900]
IC50 0.009Inhibition of recombinant human AChE using acetylthiocholine iodide as substrate by spectroscopic Ellmans method [AID600120, Type: Literature]Acetylcholinesterase [gi:113037]
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2
[SID131280900]
IC50 0.018Inhibition of Electrophorus electricus AChE using acetylthiocholine iodide as substrate by spectroscopic Ellmans method [AID600203, Type: Literature]Acetylcholinesterase [gi:14916521]
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3
[SID131280900]
IC50 0.217Inhibition of recombinant human serum BChE using butyrylthiocholine iodide as substrate by spectroscopic Ellmans method [AID600119, Type: Literature]Cholinesterase [gi:116353]
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