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CHEMBL2113424 (CID 54333857) - Compound BioActivity Data
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BioActivity Outcomes:
Active(5)
 
 
Unspecified(9)
 
 
Top Targets:
7TM GPCR Srsx(4)
 
 
 
ALBUMIN(2)
 
 
BioAssay Types:
Literature(14)
 
 
 
BioActivity Types:
Ki(5)
 
 
Data download

Chemical Probe    Active    Inactive    Inconclusive    Unspecified   

Total Bioassays: 11    Data Row: 14   Total Pages: 1   
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#SubstanceActivityBioAssayTargetLinks
OutcomeTypeValue [μM]
1
[SID163326376]
Ki 0.00403Displacement of [3H]CHA from adenosine A1 receptor of rat whole brain [AID32206, Type: Literature]Adenosine receptor A1 [gi:2827766]
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2
[SID163326376]
Ki 0.0535Binding affinity for adenosine A1 receptor was assayed by displacement of [3H]DPCPX from rat cortical membranes. [AID32012, Type: Literature]
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3
[SID163326376]
Ki 2.45Displacement of [3H]-NECA from adenosine A2 receptor of rat striatal membrane [AID33590, Type: Literature]Adenosine receptor A2b [gi:112939]
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4
[SID163326376]
Ki 2.45Displacement of [3H]-NECA from adenosine A2 receptor of rat striatal membrane [AID33590, Type: Literature]Adenosine receptor A2a [gi:8928539]
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5
[SID163326376]
Ki 4.18Binding affinity for adenosine A2A receptor was determined by displacement of [3H]-DPCPX from rat striatal membranes. [AID32863, Type: Literature]
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6
[SID163326376]
Selectivity ratio of Ki of the adenosine A2a receptor and Ki of adenosine A1 receptor [AID33948, Type: Literature]
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7
[SID163326376]
Molar potency ratio was evaluated at 37 uM [AID228923, Type: Literature]
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8
[SID163326376]
Relative binding to A2 and A1 receptors (ratio of Ki) [AID229446, Type: Literature]Adenosine receptor A2a [gi:8928539]
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9
[SID163326376]
Serum albumin binding [AID203468, Type: Literature]Serum albumin [gi:1351907]
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10
[SID163326376]
Serum albumin binding, dissociation constant [AID203472, Type: Literature]Serum albumin [gi:1351907]
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11
[SID163326376]
HPLC capacity factor (k') [AID25507, Type: Literature]
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12
[SID163326376]
Lipophilicity value was evaluated [AID28933, Type: Literature]
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13
[SID163326376]
Relative binding to A2 and A1 receptors (ratio of Ki) [AID229446, Type: Literature]Adenosine receptor A2b [gi:112939]
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14
[SID163326376]
Relative binding to A2 and A1 receptors (ratio of Ki) [AID229446, Type: Literature]Adenosine receptor A1 [gi:2827766]
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